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6,7-dimethoxy-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,2,3,4-tetrahydroisoquinoline
7-(ethanesulfonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
{7-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-5-fluoro-2,3-dihydro-1-benzofuran-2-yl}methanamine
N-cyclopropyl-5-[(2,6-difluorophenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[2-(pyridin-4-yl)ethyl]benzamide
6-methoxy-N,3-dimethyl-N-(quinoxalin-2-ylmethyl)-1-benzofuran-2-carboxamide
(2R,3R)-3-(dimethylamino)-1'-(3-fluorobenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
3-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
2-cyclopropyl-9-(1-methyl-1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1'-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(1H-indol-3-yl)pyridine-3-carboxamide
5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1-[(1R)-1-phenylethyl]-1H-imidazole
4-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)phenol
(3aR,5R,6S,7aS)-5,6-dihydroxy-N-[4-(2-methylpropoxy)phenyl]-octahydro-1H-isoindole-2-carboxamide
6-fluoro-2-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}quinolin-4-ol
4-[1-(2-methylpropyl)piperidin-3-yl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
2-tert-butyl-7,7-dimethyl-N-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-5,6,7,8-tetrahydroquinazolin-5-amine
2-({[(4-methoxyphenyl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
3,3-dimethyl-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)butanamide
1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
N-(3-methylphenyl)-3-(1-{[4-(2-oxoimidazolidin-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
2-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
1-(carbamoylmethyl)-N-[phenyl(pyridin-4-yl)methyl]piperidine-4-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}propanamide
2-(3,6-dimethylpyrazin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(furan-2-carbonyl)-4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane
4-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
N-(1,2-diphenylethyl)-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[(thiophen-2-ylmethyl)amino]benzamide
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-azabicyclo[2.2.2]octan-3-amine
2-(4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
3-[(2-{5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)sulfanyl]-4-methyl-4H-1,2,4-triazole
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)propanamide
4-[(2-chloro-4-fluorophenyl)methyl]-3-(2-oxo-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)piperazin-2-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[2-(pyridin-3-yloxy)propyl]acetamide
4-methyl-2-[1-(3-methyl-1H-indole-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
5-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-({6-chloro-3-fluoroimidazo[1,2-a]pyridin-2-yl}formamido)-N-methylbutanamide
1-ethyl-1-[2-(4-methylbenzenesulfonyl)ethyl]-3-(1-propyl-1H-pyrazol-5-yl)urea
1-(morpholin-4-yl)-3-(3-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
(7R,8aS)-7-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-{[(2R,3S,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
5-benzenesulfonamido-1-ethyl-2-methyl-N-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
(3aR,5S,6S,7aS)-2-{[4-(benzyloxy)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
3-(4-hydroxyphenyl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H-pyrazole-5-carboxamide