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N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-(2-methylphenyl)piperazin-2-one
3-{1-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
2,6-dimethoxy-N-[2-(1-methylpiperidin-3-yl)ethyl]pyrimidine-4-carboxamide
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-{4-[(3-chlorophenyl)methyl]-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-2-(2,4-difluorophenyl)ethyl)-N-methylfuran-2-carboxamide
(2E)-N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(pyridin-4-yl)prop-2-enamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[(3-methyloxetan-3-yl)methyl]amine
3-[(3R,4S)-1-[4-(aminomethyl)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(thiophen-2-yl)ethyl]pyrimidin-2-amine
3-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-ol
1-{[2-(cyclopentyloxy)phenyl]methyl}azetidin-3-ol
5-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-methyl-1,3-thiazole
9-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-diethyl-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-methylfuran-2-carboxamide
2-[4-(4-acetylphenyl)-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-benzyl-3-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(piperidin-1-yl)ethyl]benzamide
N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]pyridine-3-carboxamide
2-methoxy-1-(1'-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
N-[(5-methylpyrazin-2-yl)methyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
5-methyl-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}pyrazine-2-carboxamide
(1R,5S,6R)-3-[(3-methoxyphenyl)methyl]-N-[2-(pyridin-4-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
ethyl 1-benzyl-5-{[5-(hydroxymethyl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(5S,9aS,9bS)-5-(4-methoxy-3-methylphenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)benzamide
5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
2-{[4-(2-fluoro-6-methoxyphenyl)phenyl]sulfanyl}acetamide
4-fluoro-N-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methyl]benzamide
2-amino-N,6-dimethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrimidine-4-carboxamide
6-(dimethylamino)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-3-carboxamide
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-methylthiophene-2-carboxamide
2-[(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{3-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
3-{[2-(dimethylamino)ethyl][(4-methylphenyl)methyl]carbamoyl}benzoic acid
1-{[2-(4-ethenylphenoxy)phenyl]methyl}-4-methylpiperazine
({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)(methyl)[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amine
1-[(3-methylthiophen-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
2-(4-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
benzyl[(2-ethylpyrimidin-4-yl)methyl](oxolan-2-ylmethyl)amine
2-methyl-4-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]quinoline
8-(furan-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 4-[2-amino-3-cyano-6-(3,4-dimethylphenyl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
2-ethyl-8-{3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-2,8-diazaspiro[4.5]decan-3-one
(1R,5R)-3-methanesulfonyl-6-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane