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{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[(4-phenyl-1,3-thiazol-5-yl)methyl]amine
2-(4-acetylpiperazin-1-yl)-2-[4-(1-cyano-1-methylethyl)phenyl]acetic acid
1-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)pyrrolidin-3-amine
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
N-[2-(4-ethoxyphenyl)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
2-{2-oxo-4-[2-(oxolan-2-ylmethoxy)acetyl]piperazin-1-yl}benzonitrile
(3S,7S)-5-(2-methoxyacetyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
3-(azocan-1-yl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}propanamide
4-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-1,2-dihydrophthalazin-1-one
5-[(4-fluorophenyl)methyl]-5-[3-oxo-3-(3-propanoylpiperidin-1-yl)propyl]pyrrolidin-2-one
1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
(2E)-N-cyclopropyl-3-(3-fluorophenyl)-N-[(4-methoxyphenyl)methyl]prop-2-enamide
[4-(2-chloro-6-methoxyphenyl)pyridin-2-yl]methanol
3-[(4-acetylpiperazin-1-yl)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]ethan-1-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
(1R,2S)-N-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-2-phenylcyclohexan-1-amine
1-cyclopentyl-N5-[2-(3-fluorophenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-1-(furan-3-ylmethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-{4-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
N-{2-[(4-chlorophenyl)methoxy]ethyl}-5-cyclopropyl-1,3-oxazole-4-carboxamide
2-(4-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)phenol
4-[4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperazin-1-yl]quinazoline
4-methyl-2-{3-[2-(methylsulfanyl)ethyl]-5-{[1,2,3,4]tetrazolo[1,5-a]pyridin-6-yl}-1H-1,2,4-triazol-1-yl}pyridine
2-{4-[(4-fluorophenyl)methyl]phenyl}-2-methylpropanamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
methyl 1-benzyl-5-[(1-methoxypropan-2-yl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2R,3R)-2-methoxy-1'-[2-(thiophen-3-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
6-ethoxy-4-methyl-2-[2-(4-phenylpiperazine-1-carbonyl)pyrrolidin-1-yl]quinazoline
(3S,4S)-4-cyclopropyl-1-[2-methyl-2-(piperidin-1-yl)propyl]pyrrolidine-3-carboxylic acid
2-(dimethyl-1,3-thiazol-4-yl)-N-(thiophen-3-ylmethyl)acetamide
4-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}-2,6-dimethylphenyl acetate
N-(2,4-dimethylphenyl)-3-methyl-1H-1,2,4-triazole-5-carboxamide
5-{3H,3aH,4H,5H,9bH-cyclopenta[c]quinoline-4-carbonyl}-3-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
N-[2-(pyridin-3-yloxy)ethyl]quinoline-6-carboxamide
1-[1-(2-hydroxyethyl)piperidine-4-carbonyl]-1,4-diazepane-6-carboxylic acid
1-methyl-5-(2-phenylmethanesulfonylphenyl)-1H-1,2,4-triazole
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-ol
3-(2-chlorophenyl)-1-(2-methoxyethyl)-3-{2-[3-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-(2,3-dimethoxy-5-methylphenyl)-2-[4-(pyridin-4-yl)piperidin-1-yl]acetic acid
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-(cyclopropylmethyl)-N-propylpropanamide
5-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]-5-[(4-fluorophenyl)methyl]pyrrolidin-2-one
5-(5-methoxyfuran-2-carbonyl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{1-[(6-methoxypyridin-3-yl)methyl]piperidin-4-yl}-5-methylpyrimidine
(2H-1,3-benzodioxol-4-ylmethyl)(2,1,3-benzothiadiazol-5-ylmethyl)methylamine
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione