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2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
N-(butan-2-yl)-4-methyl-N-(3-phenylprop-2-yn-1-yl)-1,3-oxazole-5-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2R,3R)-1'-[(4-fluoro-3-methoxyphenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
N-methyl-2-({2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}amino)pyridine-3-carboxamide
4-(1H-imidazol-2-yl)-1-(2-phenylbenzoyl)piperidine
5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]pyridine-2-carbonitrile
(1S,6R)-9-(2-aminopyrimidin-4-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-(cyclopropylmethyl)-4-(5-methylpyrazine-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
2-(4-acetylphenoxy)-N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
8-[2-(morpholin-2-yl)acetyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3S,4R)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-(2-{[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}ethyl)methanesulfonamide
5-[4'-(2,2-dimethylpropyl)-3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl]-5-oxopentanamide
3-(methylsulfanyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(2-chloro-6-fluorophenyl)-N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-butyl-N-[(4-fluorophenyl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-(1,3-benzothiazol-2-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-(1H-pyrazol-1-yl)benzene-1-sulfonamide
3-(oxolan-3-yl)-5-[2-(1,1,2,2-tetrafluoroethoxy)phenyl]-1,2,4-oxadiazole
1-(cyclohexylmethyl)-N-{[4-(morpholin-4-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
7-cyclopentyl-2-(pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[2-(3,4-difluorophenyl)ethyl]-1-(furan-3-carbonyl)piperidine
N-(2-methoxyethyl)-8-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
N-[(3-methylpyridin-2-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1-{4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzoyl}piperidin-4-yl)methanol
methyl 3-(furan-3-amido)-5-({[1-(pyrrolidin-1-yl)cyclopentyl]formamido}methyl)benzoate
1-ethyl-N-[1-(1H-indol-2-yl)ethyl]-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-[1-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
3,5-dimethyl-N-(3-methyl-1-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
4-({[1-(hydroxymethyl)cyclopentyl]methyl}(methyl)amino)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N-[2-(4-fluorophenyl)ethyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
methyl (2S)-2-({5-[(2-methylpropyl)carbamoyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridin-3-yl}formamido)-3-phenylpropanoate
2-(2,5-difluorophenyl)-1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
4-(3-methyl-1H-1,2,4-triazol-5-yl)-1-[(3R,5R)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]piperidine
2,5-dimethyl-3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
8-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(4-fluorophenyl)-4-[2-(1H-imidazol-2-yl)benzoyl]-1,4-diazepane
3-(4-chlorophenyl)-5-(3,5-dimethylfuran-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[(2S)-1-[(2R,3R)-2-methoxy-3-(2-phenylacetamido)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-1-oxopropan-2-yl]acetamide
N-cyclopentyl-4-(3-fluorophenyl)-N-{[4-(oxolan-3-yloxy)phenyl]methyl}benzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
1-(2,3-dihydro-1H-indol-1-yl)-2-{10-oxo-3,9-diazaspiro[5.6]dodecan-3-yl}ethane-1,2-dione
N-(1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-(trifluoromethyl)benzamide
1-[2-(2-chlorophenyl)ethyl]-5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
5-ethyl-4-{4-[3-(3-methoxyphenoxy)azetidin-1-yl]piperidin-1-yl}-2-methylpyrimidine
2-ethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide