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5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
3-(3,4-dimethylphenyl)-N-(1,4-dioxan-2-ylmethyl)propanamide
methyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(quinoxalin-6-ylmethyl)amine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-ethyl-4-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,3-oxazole-5-carboxamide
4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-(2-ethoxyphenyl)ethan-1-one
7-(3-hydroxy-4-methoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-[(3-fluorophenyl)methyl]-6-oxo-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
ethyl 1-[2-(methylsulfanyl)pyridine-3-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{2-methyl-3-[({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1H-indol-1-yl}acetamide
5-(4-{[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
(1-{[4-(benzyloxy)-2-methoxyphenyl]methyl}pyrrolidin-3-yl)methanamine
4-hydroxy-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
[1-(naphthalene-1-carbonyl)-4-(2-phenylethyl)piperidin-4-yl]methanol
3-phenyl-1-[4-(piperidin-1-ylmethyl)benzoyl]pyrrolidin-3-ol
4-{2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl}piperazine-2-carboxylic acid
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-sulfamoylthiophene-2-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(2-phenylethyl)-3,6-diazabicyclo[3.2.2]nonane
7-(furan-3-ylmethyl)-N-methyl-N-(oxan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
3-(1H-1,3-benzodiazol-2-yl)-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]propan-1-one
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-(1-phenylethyl)benzamide
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-methyl-1,4-diazepane
1-(3-cyclopropyl-1H-1,2,4-triazole-5-carbonyl)-2-methyl-2,3-dihydro-1H-indole
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amine
N-[(4-hydroxyazepan-4-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
4-{[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
2,2-diphenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
(1S,4S)-2-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-azabicyclo[2.2.1]heptane
methyl (2S,4R)-4-[2-(1H-pyrazol-1-yl)benzamido]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxylate
(3S,9aR)-8-[(5-methylthiophen-2-yl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,2-dimethylpiperazine
2-[1-(furan-3-ylmethyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-yl]ethan-1-ol
N-(pyridin-4-ylmethyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}cyclopropanamine
4-(3-fluorophenoxy)-1-(3-fluoropyridin-2-yl)piperidine-4-carboxylic acid
4-methoxy-N-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
4-(3-chlorophenoxy)-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(naphthalen-2-yl)ethyl]-1,3-oxazole-4-carboxamide
5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(1-methyl-1H-pyrrol-3-yl)-N-(oxolan-2-ylmethyl)acetamide
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylate
ethyl 2-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetate
N-(3-chloro-4-methoxyphenyl)-6-(3,4-dimethylbenzoyl)-6-azaspiro[2.5]octane-1-carboxamide
1-(butan-2-yl)-N3-[(5-chlorothiophen-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(4aR,8aR)-4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-2H-1,4-benzoxazine