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2-amino-7-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
2-chloro-4-({3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
(1R,5R)-N,N-dimethyl-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2,3-dioxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
2-benzyl-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}morpholine
9-[(5-chlorothiophen-2-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
N-(5-hydroxypentyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-cyclohexyl-3-[2-(morpholin-4-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-[1-(3-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
2-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanamide
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine
4-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-7-methyl-3,4-dihydro-2H-1,4-benzothiazin-3-one
1-[cyclohexyl(methyl)amino]-3-{4-[(cyclopentylamino)methyl]-2-methoxyphenoxy}propan-2-ol
N-[(2R,3R)-2-(benzyloxy)-1'-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
[(3-{[1-(2-cyclopropylquinoline-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(1,3-thiazol-2-ylmethyl)amine
[1-(2-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)piperidin-3-yl]methanol
1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3-propylpiperidine-3-carboxylic acid
5-(4-chloro-3,5-dimethylphenoxymethyl)-3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazole
N'-(2,5-dimethylphenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanediamide
2-fluoro-N-({7-[2-(3-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
5-(2-chlorophenyl)-2-methyl-N-[(3-methylpyridin-2-yl)methyl]furan-3-carboxamide
2-methyl-2-{4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}propanenitrile
4-(pyrimidin-2-yl)-1-(quinoline-3-carbonyl)piperazine-2-carboxylic acid
N-[4-(3-methoxyphenyl)phenyl]-1-(pyridine-4-carbonyl)piperidine-3-carboxamide
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[1-(2-phenylethyl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(3-methylthiophen-2-yl)methyl]({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})(pyridin-2-ylmethyl)amine
3,5-dimethyl-4-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-pyrazole
1-[1-(cyclobutylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-methyl-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,3-benzothiazole
N-{1-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
3-methyl-8-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}-1H-pyrazole-3-carboxylic acid
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
N-[(2R,3R)-1'-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-1-methylpiperidine-4-carboxamide
(1S,5R)-3-(2-methoxypyridine-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopentyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)cyclohexanecarboxamide
2-(dimethylamino)-2-(2-methylphenyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}acetamide
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
5-{[(1-methylpiperidin-4-yl)(2-phenylethyl)amino]methyl}-1,2,4-oxadiazole-3-carboxamide
1-(azepan-1-yl)-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-(2,3-dihydro-1H-indene-5-carbonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-(2,5-dioxoimidazolidin-1-yl)-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]acetamide
2-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-N,N,5-trimethylpyrimidin-4-amine
1-(2-cyclopropylpyrimidine-5-carbonyl)-N-(furan-2-ylmethyl)piperidine-4-carboxamide
2-(1H-1,2,4-triazol-1-ylmethyl)-5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]pyrimidin-4-ol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(methylamino)pyridine-4-carboxamide