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2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethan-1-one
5-(1-benzofuran-2-yl)-N-(1-benzylpyrrolidin-3-yl)-1,2,4-triazin-3-amine
7-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)-2,7-diazaspiro[4.5]decane
N-(2,6-dimethylpyridin-3-yl)-4-(2-methoxyphenoxy)piperidine-1-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
(4aR,8aS)-1-[2-(2-fluorophenyl)ethyl]-6-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
2-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzonitrile
3-{5-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(propan-2-yl)propanamide
3-({4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
4-(2-{1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}ethyl)morpholine
N-propyl-2-{pyrazolo[1,5-a]pyridin-7-yl}benzamide
N-[(1-methylpiperidin-3-yl)methyl]-9-oxo-9,10-dihydroacridine-4-carboxamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
[(2S)-1-(3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-2-yl]methanol
1-[(2-methoxyphenyl)methyl]-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
(1-benzothiophen-2-ylmethyl)({4-[(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)methylamine
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
2-(4-{[(2-amino-5-ethylpyrimidin-4-yl)(methyl)amino]methyl}piperidin-1-yl)ethan-1-ol
3-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-5-[2-(piperidin-2-yl)ethyl]phenol
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-(pyridin-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(6-methylpyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-1-phenylcyclopropane-1-carboxamide
N-cyclopentyl-4-(2-methyl-1H-imidazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{4-phenyl-1-[2-(pyridin-2-yl)ethyl]piperidin-4-yl}ethan-1-one
1-(3,5-dimethylfuran-2-carbonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-N-methylpyrimidin-2-amine
N'-(2-ethoxyphenyl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]propanediamide
2-[1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyrimidine-4-carbonyl)piperidin-3-ol
3-(2-chloro-4-fluorobenzoyl)-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-cyclopropyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
3-(2-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-2-oxoethyl)-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-8-fluoro-N-methylquinoline-2-carboxamide
1-{2-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propyl}-3,5-dimethyl-1H-pyrazole
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
1-[2-(pyridin-3-yl)-4-{[(1r,4r)-4-hydroxycyclohexyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-methyl-9-(4-phenyl-1,3-thiazole-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
N-(1-benzothiophen-2-ylmethyl)-N-methyl-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-[2-(1H-pyrazol-1-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
[(2-fluoro-4,5-dimethoxyphenyl)methyl](methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-({8-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide
N-cyclopropyl-5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-4-methylpiperazin-2-one
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-[(3-methoxyphenyl)methyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
[1-({[2-(propylsulfanyl)pyrimidin-5-yl]methyl}amino)cyclopentyl]methanol
4-{1-benzyl-5-[2-(2-chlorophenyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
1-[(2-methoxyphenyl)methyl]-4-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine