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N-(3-{[3-(naphthalene-2-carbonyl)piperidin-1-yl]sulfonyl}phenyl)acetamide
1-methyl-N-({5-methyl-2-[3-(pyridine-4-amido)phenyl]-1,3-oxazol-4-yl}methyl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
methyl 6-(2-{[4-(thiophen-2-yl)butanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
2-chloro-3-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]urea
2-[4-(4-cyclopentylpyrimidin-2-yl)-1-methylpiperazin-2-yl]ethan-1-ol
(3R,4R)-4-cyclopropyl-3-methyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-ol
N-(3-hydroxy-2,2-dimethylpropyl)-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-[(4-methoxypyridin-2-yl)methyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
ethyl 1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-phenoxyacetamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
1-(1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)ethan-1-one
6-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-1H-indole
5-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-1-(propan-2-yl)-1H-imidazole
N-[(1-ethylpiperidin-3-yl)methyl]-N-methyl-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-[2-(thiophen-2-yl)ethyl]benzamide
1-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-2-methoxyethan-1-one
1-(4,7-dimethylquinazolin-2-yl)-N-[(1S)-1-phenylethyl]piperidine-3-carboxamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2,5-dimethoxyphenyl)methyl]propanamide
4-hydroxy-2-{[(2-hydroxyethyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}quinoline-6-carboxamide
(3R,4R)-1-[(5-fluoro-2-methoxyphenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
[1-(5-{[ethyl(methyl)sulfamoyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N-(3-hydroxy-3-phenylpropyl)-N-methyl-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-({7-[2-(3,4-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
1-{4-[3-({[2-(3-methoxyphenyl)ethyl]amino}methyl)-7-(methylsulfanyl)quinolin-2-yl]piperazin-1-yl}ethan-1-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethan-1-one
N-(3-hydroxypropyl)-1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
2-(methoxymethyl)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-({3-[3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
6-methyl-3-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-{3-oxo-3-[3-(pyridine-3-carbonyl)piperidin-1-yl]propyl}pyrrolidin-2-one
1-methyl-5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-1-yl)-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
N2,N2,5,6-tetramethyl-N4-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidine-2,4-diamine
2-ethyl-4-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1H-imidazol-2-yl}pyrimidine
3-[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-N-cyclopropylpropanamide
8-[2-(dimethylamino)benzoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-cyclopropyl-8-(3-ethoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[1-(4,6-dimethylquinazolin-2-yl)piperidin-4-yl]amino}butan-2-ol
1-(4-chloro-2-methoxy-5-methylphenyl)-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
N-({1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-3-yl}methyl)furan-2-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
7-(2-cyclohexylethyl)-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
4-(4-chlorophenoxy)-N-(2,2-difluoroethyl)piperidine-4-carboxamide