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N-(1-butyl-1H-pyrazol-5-yl)-4-[(3-oxopiperazin-1-yl)methyl]benzamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[(3-methylpyridin-2-yl)methyl]propanamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(pyrrolidin-1-yl)pyridine
8-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-methyl-2-(3-methylphenoxy)-1-[3-(pyridin-3-yl)azetidin-1-yl]butan-1-one
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)-3-(trifluoromethyl)benzene-1-sulfonamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-ethyl-8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-[2-(3-chlorophenyl)ethyl]-4-[(4,4,4-trifluorobutyl)amino]pyrrolidin-2-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-indol-3-yl)acetamide
2-{1-[(2-fluorophenyl)methyl]-4-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(4aS,8aS)-2-[2-(4-methoxyphenoxy)ethyl]-decahydroisoquinoline
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}propanamide
8-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{2-methoxy-5-[2-(1H-pyrazol-1-yl)propanamido]phenyl}benzamide
2,5-dimethoxy-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-(1,3-benzothiazol-2-yl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
2-{1-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
N,5-dimethyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}pyrazine-2-carboxamide
1-ethyl-3-(2-methylphenyl)-3-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(1-phenyl-1H-pyrazol-4-yl)-1H-1,2,3-triazole
3-ethyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}urea
1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-4-(pyridin-3-yl)piperazine
(4aS,7aR)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 9-[2-(2-fluorophenyl)ethoxy]-7-oxo-3-[(1R,2S)-2-propylcyclopropanecarbonyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(3-{[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
1-[4-({[3-(difluoromethoxy)phenyl]methyl}amino)-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-fluoro-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-butyl-5-[1-(2-fluorophenyl)cyclopropyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
(3aR,7aS)-2-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2,2-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}butanamide
N-(propan-2-yl)-2-[(2,4,6-trimethylphenyl)formamido]acetamide
5-(dimethylamino)-2-{2-oxo-2-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
(4aS,7aR)-1-[(2,5-dimethylphenyl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,5S,6R,7S)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-[1-(pyrimidin-4-yl)ethyl]pyrimidine-5-carboxamide
2-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-6-methylpyridine
methyl (2S,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
2-methyl-5-[3-(piperidin-1-yl)pyrrolidine-1-carbonyl]phenol
1-ethyl-8-(1H-indol-3-ylmethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}acetamide
N-{[4-(methylsulfanyl)phenyl]methyl}-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
5-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-[(3,4,5-trimethoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
ethyl 2-(1-{[4-(4-acetyl-1,4-diazepan-1-yl)quinazolin-2-yl]methyl}piperidin-2-yl)acetate
(2-{[4-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperazin-1-yl]methyl}phenyl)methanol