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(2S)-4-methyl-2-phenyl-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(3-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-yl)acetamide
1,3,5-trimethyl-4-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
N-({1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]azetidin-3-yl}-2-methylpiperidine
N-{1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
2-cyclopropyl-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-{[7-(2,3-dimethylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
8-(6-ethyl-2-methylquinoline-4-carbonyl)-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
5-[1-cyclohexyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
N-{[3-methyl-7-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-carboxamide
2-(4-hydroxypiperidin-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
N-[4-(3-fluorophenyl)phenyl]-1-[2-(methylsulfanyl)acetyl]piperidine-3-carboxamide
methyl 4-{[10-(3-hydroxypiperidine-1-carbonyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-3-yl]methyl}benzoate
N-({3-methyl-7-[2-(naphthalen-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(pyrimidin-2-ylsulfanyl)acetamide
4-(5-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)quinoline
(1-benzofuran-2-ylmethyl)(methyl)(oxan-2-ylmethyl)amine
N-(furan-3-ylmethyl)-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(4-chlorobenzoyl)piperidin-1-yl]propan-1-one
(3S)-N,N-dimethyl-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)azepan-3-amine
(3aS,6aS)-2-(ethanesulfonyl)-5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-benzyl-3-(pyridin-2-ylmethyl)-8-(quinolin-7-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-{4-[(1,4-dioxan-2-ylmethyl)amino]piperidin-1-yl}phenyl)-5-phenylpentanamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(pyridin-2-yl)propan-2-yl]propanamide
2-chloro-4-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenol
ethyl 1-(3-methoxypropanoyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-3-carbonitrile
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
2-oxo-N-(1-phenylbutyl)-2H-pyran-5-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methyl-1,3-oxazole-4-carboxamide
3-phenyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
(2S,4R)-4-(dimethylamino)-N-[2-(4-fluorophenyl)ethyl]-2-(hydroxymethyl)pyrrolidine-1-carboxamide
4-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(4-sulfamoylphenyl)methyl]acetamide
3-{[(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
8-[(2E)-4-methylpent-2-en-1-yl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-[(4-methoxyphenyl)methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]piperidine-4-carboxylate
3-{3-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridine
1-phenyl-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclopropane-1-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[5-(4-methoxyphenyl)furan-2-carbonyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)-4-(2-oxopyrrolidin-1-yl)benzamide
ethyl 1-{6-[4-(methylsulfanyl)phenyl]-3-(thiomorpholine-4-carbonyl)pyridin-2-yl}piperidine-4-carboxylate