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N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-6-oxo-1-(prop-2-en-1-yl)piperidine-3-carboxamide
methyl 9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-3-(3-methylfuran-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(3-methylphenoxy)-1-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
1-[2-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(pyridin-2-yl)pyrrolidin-3-yl]methanol
3-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-3-yl}benzoic acid
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
8-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 6-{2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyrimidine-4-carboxylate
2-(propan-2-yl)-4-(1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-imidazol-2-yl)pyrimidine
2-fluoro-5-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]phenol
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(pyridin-4-yl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxamide
3-[(3-methylbutyl)amino]-N-(thiophen-2-ylmethyl)propanamide
2-[5-(4-methanesulfonylphenyl)-4-phenyl-1H-imidazol-1-yl]acetamide
[1-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-yl]methanol
2-(diethylamino)-1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
4-chloro-3-({[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
7-(8-chloroquinolin-2-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
{[5-(ethanesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(methyl)[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-[7-(3-acetylpiperidine-1-carbonyl)-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
1-methyl-4-[2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetyl]piperazin-2-one
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)(pyridin-3-ylmethyl)amine
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-cyclobutanecarbonyl-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 5-{[(2-methylphenyl)methyl]amino}-1-(2-methylpropyl)-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-methyl-3-({4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}methyl)-4H-chromen-4-one
2-(2-fluorophenoxymethyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyrazin-2-yl)ethan-1-one
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-methoxyphenyl)methyl]-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
4-[(2-chlorophenyl)methyl]-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
6-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyridine-2-carboxylic acid
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-methylfuran-2-carboxamide
methyl 4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]benzoate
N-[2,5-dimethyl-3-({3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1H-pyrrol-1-yl]acetamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}propan-1-one
ethyl 1-(3-chlorobenzoyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
(2E)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
2-methyl-N-{2-[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
4-(2-methoxy-2-phenylacetyl)-1-(2-methylphenyl)piperazin-2-one
2-(3-methoxypropyl)-9-[4-(trifluoromethyl)pyrimidin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-benzothiophen-2-ylmethyl)-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(dimethyl-1,3-oxazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-N-({4-methoxy-3-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-2,2-diphenylacetamide
3-(but-2-yn-1-yl)-5-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
2-(1H-imidazol-2-yl)-N-[2-(pyridin-2-yl)ethyl]benzamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-N-(2-phenylethyl)piperidine-4-carboxamide
1-[(4aR,8aS)-6-benzoyl-decahydro-1,6-naphthyridin-1-yl]-2-(methylsulfanyl)ethan-1-one