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5,6-dimethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrimidin-4-amine
1-[2-(morpholin-4-ylmethyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-benzoyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]piperidin-4-amine
N-cyclopropyl-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-phenylethane-1,2-dione
1-cycloheptyl-6-oxo-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-{[7-(3-chlorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
3-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)sulfamoyl}-N,N-dimethylbenzamide
N-[6-methoxy-2-oxo-4-(1,3-thiazol-2-yl)-1,2,3,4-tetrahydroquinolin-7-yl]furan-2-carboxamide
1-[(4aR,8aS)-1-(2-methyl-1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(4-methoxyphenyl)ethan-1-one
4-(1H-imidazol-2-ylmethyl)-3-propylmorpholine
(1S,4S)-2-{4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-2-azabicyclo[2.2.1]heptane
ethyl 4-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazine-1-carboxylate
5-(1H-imidazol-2-yl)-1-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-phenyl-1H-imidazole
6-(5,6-dimethylpyrimidin-4-yl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
4-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}pyridine
[1-(2-methoxyphenyl)ethyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
8-(5-methyl-1,3-benzoxazol-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-N-methyl-1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxamide
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(5S)-5-{[5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyrrolidin-2-one
N-{[3-methyl-7-(5-methylthiophene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}pyrazine-2-carboxamide
N-{4-[5-methyl-4-({[(1R,2S)-2-propylcyclopropyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}pyridine-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-fluoro-1H-indol-2-yl)methyl]acetamide
2-[3-cyclopropyl-5-({[2-(pyrrolidin-1-yl)ethyl]sulfanyl}methyl)-1H-1,2,4-triazol-1-yl]pyridine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)acetamide
8-[(3,4-dimethoxyphenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(2-fluorophenyl)-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2,4-triazin-3-amine
1-[(3,4-dimethylphenyl)methyl]-4-(4-hydroxy-2-methylpyrimidine-5-carbonyl)piperazin-2-one
3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(1,4-dioxan-2-ylmethyl)propanamide
1-methyl-4-(quinoxaline-5-carbonyl)-1,4,9-triazaspiro[5.5]undecane
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-amino-3-(3,4-dimethoxyphenyl)propan-1-one
(2S,4R)-N-ethyl-4-[2-(pyridin-4-yl)acetamido]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
N-[(3R,4S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-hydroxypropanamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
2-(4-{[1-(cyclopropylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
3-[2-(9H-fluoren-2-yl)-1H-imidazol-1-yl]-2,3-dihydro-1λ6-thiophene-1,1-dione
3-[(3-chlorophenyl)methyl]-N-(2,2-dimethyloxan-4-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[1-(furan-2-yl)ethyl]-N-methylpiperidine-3-carboxamide
4-{[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzoic acid
N-[2-(dimethylamino)ethyl]-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
1-[(2-fluorophenyl)methyl]-N-[2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2,8-dimethyl-4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]quinoline
1-{[3-(4-fluorophenoxy)phenyl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-methyl-1H-pyrazol-1-yl)acetamide
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-3-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
3-[2-(methylsulfanyl)benzoyl]-1-(prop-2-ene-1-sulfonyl)piperidine
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one