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N-cyclopropyl-4-{[2-(oxan-3-yl)ethyl]sulfamoyl}benzamide
1-(4-{[3-(4-ethylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-3-methoxyphenyl)ethan-1-one
methyl(1H-pyrazol-3-ylmethyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
1-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-3,3-dimethylurea
2-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-dihydroquinoline-3-carboxamide
4-{3-[3-(3-methylphenoxy)azetidine-1-carbonyl]phenyl}morpholine
2-{1-[(4-methylphenyl)methyl]-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-2-methylpiperidine
3-(cyclopropylmethyl)-5-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
3-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
2-(morpholin-4-ylmethyl)-4-(2-phenylethyl)-1,4-oxazepane
2-(2-methoxyphenyl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine
4-ethyl-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{3-[4-(cyclopentylmethyl)piperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-fluoro-N-(4-{4-[(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
3-ethyl-4-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1H-pyrazole-5-carboxamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopent-1-ene-1-carboxamide
3-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}sulfonyl)benzonitrile
6-cyclopentyl-2-(3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-cyclopentyl-4-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
6-methyl-2-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)pyrrolidine-2,5-dione
1-[7-(6,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
2-(4-acetylphenoxy)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
4-(3-hydroxy-3-methylbutyl)-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]benzamide
1-(1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
5-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridine-2-carbonitrile
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(9H-purin-6-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[5-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
methyl(4-methyl-1-phenylpentyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
1-(carbamoylmethyl)-N-methyl-N-[(4-phenoxyphenyl)methyl]piperidine-3-carboxamide
(1R,2S)-1-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2,3-dihydro-1H-inden-2-ol
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
7-(2-methyl-1,3-thiazole-4-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[3-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-(1-benzofuran-5-ylmethyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
4-(2,6-difluoro-3-methoxybenzoyl)-2-ethyl-1-(propan-2-yl)piperazine
methyl 7-oxo-3-[2-(phenylsulfanyl)acetyl]-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-benzyl-9-[(2R)-2-cyclohexyl-2-hydroxyacetyl]-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-N-[(1-ethyl-1H-indazol-3-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-{1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-{1-[7-(2-cyclohexylacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-(dimethylamino)acetamide
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-4,6-dimethylpyridine-3-carbonitrile
1-(4-chlorophenyl)-N-({1-[(2-hydroxyphenyl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
2,5-dimethoxy-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-N,N-diethylpyrrolidin-3-amine