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{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
2-(dimethylamino)-4-methyl-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidine-5-carboxamide
7-(cyclopropylmethyl)-2-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
(3R,4S)-1-(dimethyl-1,3-oxazole-5-carbonyl)-4-propylpyrrolidin-3-amine
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-4-carboxamide
methyl 4-(5-methyl-4-{[methyl(quinoxalin-6-ylmethyl)amino]methyl}-1,3-oxazol-2-yl)benzoate
2,6-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidine-4-carboxamide
2-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-3-yl)propan-2-ol
3-({2-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-[(3-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-phenyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1H-1,2,3-triazole-4-carboxamide
4-(2-cyclopropylquinoline-4-carbonyl)-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-methyl-3-phenylpiperidine
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-6-methylpyridine-2-carboxamide
1-[(2-fluorophenyl)methyl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-oxopiperidine-3-carboxamide
7-[(4-methoxy-2,5-dimethylphenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(2-methoxyethyl)methylamine
N-[(2S,4R,6S)-2-(2-cyanophenyl)-6-(2-phenylethyl)oxan-4-yl]acetamide
4-(1-butyl-1H-imidazol-2-yl)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidine
(2S,4R)-4-[4-({[(6-chloropyridin-3-yl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
1-[5-methoxy-2-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
N-methyl-5-{[2-(5-methylfuran-2-yl)phenyl]methyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 5-{[(3,4-dimethoxyphenyl)methyl]amino}-3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-(2-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-4-fluorophenyl)-1H-pyrazole
3-methyl-N-{1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
2-(6-methyl-1-benzofuran-3-yl)-N-(1,2-oxazol-3-yl)acetamide
4-{1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-3-yl}benzoic acid
5-cyano-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-(oxolan-2-ylmethyl)-1-[1-(thian-4-yl)piperidin-4-yl]piperidine-4-carboxamide
N,N-diethyl-1-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]piperidine-3-carboxamide
ethyl 2-[4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)morpholin-3-yl]acetate
N-cyclopropyl-1-[1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
4-({1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}methyl)morpholine
(3S,4S)-4-(4-fluorophenyl)-1-(1H-indazole-3-carbonyl)piperidin-3-ol
[(2S,4R)-1-methyl-4-{[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]amino}pyrrolidin-2-yl]methanol
(3R,4R)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-(furan-2-ylmethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl})amine
N-cyclopropyl-3-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)propanamide
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-5-methoxyfuran-2-carboxamide
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
1-(furan-2-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(5-oxopyrrolidin-2-yl)acetamide
3-(2,3-dihydro-1H-inden-2-yl)-5-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
N-{2-[(pyridin-3-yl)amino]ethyl}-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
5-methyl-1-(4-methylphenyl)-4-[4-(pyrrolidin-1-yl)butanoyl]piperazin-2-one