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2-{1-[(3,4-difluorophenyl)methyl]-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[3-(2-methylphenoxy)azetidin-1-yl]-2-(propylsulfanyl)ethan-1-one
4-[3-(aminomethyl)pyrrolidine-1-carbonyl]-N-(pyridin-4-ylmethyl)aniline
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
(2R,3R)-3-amino-1'-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}benzoic acid
N-{[7-(3-chlorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(1H-imidazol-1-yl)acetamide
(3R,4R)-1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-(methoxymethyl)pyrrolidine
N-[(1S,2R)-2-(cyclooctylamino)cyclobutyl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide
5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(furan-2-yl)pyrrolidine
N-(2-methoxyethyl)-3-methyl-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
N-cyclopropyl-1-[1-(pyrazin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
({4-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-yl}methyl)dimethylamine
2,6-difluoro-N-{[7-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
N-cyclopropyl-1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-[1-ethyl-5-(1-phenylcyclopropanecarbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,6-dimethyl-2-oxo-2H-pyran-5-carboxamide
N,5-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-[(2R,3R)-1'-(4-acetamidobenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
2-({6-[6-(benzyloxy)pyridin-3-yl]pyridazin-3-yl}(methyl)amino)ethan-1-ol
N-{2-methyl-1-oxo-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propan-2-yl}thiophene-2-carboxamide
5-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-ethyl-4-methyl-1,3-oxazole
(4aS,8aR)-1-butyl-6-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]pyridazine
(3S,4S)-4-cyclopropyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-(2,4-dimethylphenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(methylamino)pyridine-4-carbonyl]pyrrolidin-3-yl]acetamide
1-[4-(2,3-dimethylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-phenylpropan-1-ol
N-cyclopentyl-6-ethyl-2-(pyrimidin-5-yl)quinoline-4-carboxamide
2-chloro-N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)pyridine-4-carboxamide
3-cyclopropyl-5-[2-(4-methylbenzenesulfonyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
(3aR,6aR)-2-(cyclobutylmethyl)-5-[(5-methylpyrazin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
3-{[(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
3-(2,3-dihydro-1H-inden-2-yl)-5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]quinoxaline
N-(2,3-difluorophenyl)-2-(2-hydroxyethyl)pyrrolidine-1-carboxamide
1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
ethyl 4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazine-1-carboxylate
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-hydroxypropyl)acetamide
4-(2-fluorophenoxy)-1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
6-[(3R,5R)-5-(morpholine-4-carbonyl)piperidine-3-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
4-(1H-imidazol-2-yl)-1-[3-(piperidin-3-yl)benzoyl]piperidine
2-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
1-[(4-chlorophenyl)methyl]-N-(2-hydroxyethyl)-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide