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5-hydroxy-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyrazine-2-carboxamide
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-3-ene-1-carboxamide
methyl 4-[(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]benzoate
2-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}-1H-1,3-benzodiazole
1-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}ethan-1-one
N,N-diethyl-1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-{1-oxaspiro[4.5]decan-3-yl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-amino-4-(isoquinolin-5-yl)-6-(1-methyl-1H-pyrrol-2-yl)pyridine-3-carbonitrile
8-[(2,4-difluorophenyl)methyl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({5-[(4-fluoro-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
5-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
1-cyclopropanecarbonyl-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
methyl (2S)-2-({1-[4-(2,4-dimethylbenzamido)phenyl]piperidin-4-yl}amino)-3-methylbutanoate
N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]cyclopropanesulfonamide
1-(1H-imidazol-4-ylmethyl)-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
4-[(4-methoxyphenyl)methyl]-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aR,7aS)-1-cyclopropanecarbonyl-4-(1-propyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(trimethyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-benzyl-N-methyl-2-(piperazine-1-carbonyl)-2,3-dihydro-1H-inden-2-amine
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-(1H-pyrrole-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(2R,3R)-1'-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3,3-dimethylbutanamide
methyl 2-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]benzoate
1-methyl-3-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
4-cyclobutyl-2-(4-ethylpiperazin-1-yl)-6-methylpyrimidine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-methyloxetane-3-carbonyl)pyrrolidine-3-carboxylic acid
5-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
(1s,4s)-4-({2-[(4-methoxyphenyl)methyl]morpholin-4-yl}methyl)cyclohexan-1-amine
2-(1H-imidazol-2-yl)-N-[(2S)-1-methoxypropan-2-yl]benzamide
1-(5-fluoro-1H-indole-2-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(4-benzylpiperazine-1-carbonyl)-6-[(2,4,5-trimethoxyphenyl)methyl]-6-azaspiro[2.5]octane
N,N-dimethyl-3-[3-(oxolan-3-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]aniline
2-(2,5-dimethoxyphenyl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methylpyrimidin-2-amine
N-(2-hydroxyethyl)-5-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1S,3R)-3-amino-N-[(3-methoxy-2-propoxyphenyl)methyl]cyclopentane-1-carboxamide
2-{2-[1-(6-chloroquinolin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one
1-(4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-pyrazole
3-{1-[1-(2,4-difluorobenzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-[2-(diethylamino)ethyl]-5-(4-methoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(2-methoxyethoxy)ethan-1-one
(2S)-2-amino-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]propan-1-one
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
[(1-cyclopentylpiperidin-4-yl)methyl][(8-methoxyquinolin-2-yl)methyl](pyridin-3-ylmethyl)amine
3-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-1-methyl-1-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea