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5-[1-(3-chloro-4-fluorobenzoyl)piperidin-4-yl]-5-(2-methylpropyl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
N-[(3-fluoro-4-methylphenyl)methyl]-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
1-[(1-benzylpiperidin-3-yl)methyl]-3-(3-cyano-4-methoxyphenyl)urea
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(6-hydroxy-6-methylheptan-2-yl)-1-(5-methoxy-2-methylphenyl)urea
[4-(3-phenylpropyl)piperidin-4-yl]methanol
3-ethyl-8-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-2-methyl-4-phenylpiperazine
1-[2-hydroxy-3-(3-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
2-amino-6-(5-chlorothiophen-2-yl)-4-(1-ethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-methyl-6-[1-(pentan-2-yl)-1H-imidazol-2-yl]pyridine
N-[(3R,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-(cyclohex-3-ene-1-carbonyl)-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-(pyrrolidin-1-yl)ethan-1-one
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]-N-(3-chloro-4-methoxyphenyl)propanamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidine
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-N-[(3-chlorophenyl)methyl]propanamide
3-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-2-yl}propanoic acid
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
3-[4-(3-cyclopentyl-1-ethyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-1λ6-thiolane-1,1-dione
2-{[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
1-(5-methyl-2H-1,2,3-triazole-4-carbonyl)-4-(oxan-4-yl)-1,4-diazepan-6-ol
3-chloro-2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-indole
2-[3-(dimethylamino)propyl]-9-(5-ethyl-1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[6-(5-chloro-2-methoxypyridin-4-yl)pyridin-3-yl]methyl}acetamide
8-(2-amino-2-methylpropanoyl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one
(5S,9aS,9bS)-5-(6-chloro-2H-1,3-benzodioxol-5-yl)-2-(2,3-dihydro-1H-inden-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{[5-(5-chloropyridine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(furan-3-ylmethyl)methylamine
1-(3-methanesulfonamidophenyl)-3-[2-(morpholin-4-yl)ethyl]urea
4-(1,3,7-trimethyl-1H-indole-2-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-(4-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}phenoxy)acetic acid
3-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-oxoethyl)-5,7-dimethyl-2,3-dihydro-1H-indol-2-one
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-2-methylpiperidine
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-propyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
methyl (2S,4R)-1-[2-(2,2-dimethylpropanamido)-5-methylthiophene-3-carbonyl]-4-hydroxypyrrolidine-2-carboxylate
2-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyridine-4-carboxamide
2-{2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
6-[2-(1,3-benzothiazol-2-yl)pyrrolidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
(2R)-1-[(4,8-dimethoxynaphthalen-1-yl)methyl]pyrrolidine-2-carboxamide
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
N-(2-methylphenyl)-7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-{5-[1-(2-cyclohexylethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
2-amino-4-(2-aminopyrimidin-5-yl)-6-(6-methoxynaphthalen-2-yl)pyridine-3-carbonitrile
3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-7-methyl-1,2-dihydroquinolin-2-one
1-(2-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-2-methylpropanamide
5-cyclopropanecarbonyl-1'-[(2-fluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4,5,6,7,8-octahydroquinolin-2-one
2-(2-methyl-1H-indol-3-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one