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N-ethyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
4-(1H-1,3-benzodiazol-1-yl)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
1-(oxan-4-yl)-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
8-(2-ethylpyridine-4-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(dimethylamino)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(2-methylphenyl)acetamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}acetamide
5-{2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-[(3R,4R)-4-hydroxypiperidin-3-yl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-{[3-(ethoxycarbonyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
N-cyclohexyl-6-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
N-tert-butyl-2-(4-{[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl}phenoxy)acetamide
7-(2,3-dimethoxyphenyl)-9-methoxy-4-(4-phenylbutan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3S,5S)-1-benzyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
8-(butan-2-yl)-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
2-{3,5-dimethyl-4-[(1R,2R)-2-phenylcyclopropaneamido]-1H-pyrazol-1-yl}acetic acid
methyl 6-(3-fluorobenzoyl)-2-[(4-fluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[1-(5-chloro-2-methoxyphenyl)-5-[3-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl]acetamide
(3R,9aR)-8-(2,5-difluorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(pyrimidin-4-yl)ethyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-{1-[2-(piperidin-1-yl)acetyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
4-[2-(pyrrolidin-3-yl)benzoyl]piperazine-1-carboxamide
1-(cyclohexylmethyl)-N3-cyclopropyl-4-oxo-N5-[phenyl(pyridin-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-{4-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
3-ethoxy-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propan-1-one
2-amino-4-[5-(oxan-2-yl)thiophen-2-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
methyl 2-chloro-4-({[3-(morpholin-4-yl)propyl]carbamoyl}amino)benzoate
7-cyclobutaneamido-N,1-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(1S,2R)-N1-butyl-N1-ethyl-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-3-(5-methylfuran-2-yl)-1H-pyrazole
N-[2-(dimethylamino)-2-(4-fluorophenyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(1-methyl-1H-imidazol-2-yl)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidine
4-(2,1,3-benzothiadiazol-5-ylmethyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
6-[1-(3-chloro-2-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-cyclopropyl-N'-(2,4-dimethylphenyl)-N-[(2-methoxyphenyl)methyl]propanediamide
3-chloro-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pyridin-2-amine
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
2-{2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
4-(4-chlorophenoxy)-N-ethyl-N-(oxan-4-yl)piperidine-4-carboxamide
5-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-methyl-4-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-4-phenylpiperidine
N-ethyl-5-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]pyrimidin-2-amine
(2S,4S)-4-(4-cyanobenzamido)-1-(cyclopentylmethyl)-N-ethylpyrrolidine-2-carboxamide
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
N-(2-ethyl-4-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)acetamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
dimethyl[2-({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(thiophen-3-ylmethyl)amino)ethyl]amine