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1-cyclobutanecarbonyl-4-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,4-diazepane
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3-(5-methylfuran-2-yl)-1H-pyrazole
2-[1-(thiophen-2-ylmethyl)-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-4H-chromen-4-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-{1-methyl-4-[(2,4,6-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]acetamide
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]-N-(5-chloro-2-methoxyphenyl)propanamide
4-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}-2-(1H-1,2,3,4-tetrazol-1-yl)pyridine
1-{[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})carbamoyl]methyl}piperidine-4-carboxamide
5-(2-methoxyphenyl)-1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
7-(5-ethyl-1,3-oxazole-4-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4-methylphenol
4-({1-[3-(piperazin-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
3-(3-fluorophenyl)-N-[(3-hydroxypiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-(2-{1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N,2-dimethyl-4-oxo-N-(quinolin-5-ylmethyl)-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-(3-phenylpropyl)-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
(3R,7S,8aS)-7-{[(2-chlorophenyl)methyl]amino}-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}phenyl)methanol
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
3-[2-amino-4-(4-cyclopentyl-3-oxopiperazin-1-yl)-6-methylpyrimidin-5-yl]propanoic acid
2-(2,3-dimethoxyphenyl)-1-{1-oxaspiro[4.4]nonan-3-yl}-1H-imidazole
(benzylsulfamoyl)(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[(3-fluorophenyl)methyl]methylamine
3-[5-(2-methoxy-2-phenylacetyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-[(3-chlorophenyl)methyl]-1-(9H-purin-6-yl)piperidine-3-carboxylic acid
1-[(1-{6-[(1-hydroxy-3-methylbutan-2-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-{[(1-hydroxybutan-2-yl)(pyridin-2-ylmethyl)amino]methyl}benzoic acid
2-(1H-1,2,4-triazol-3-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}benzamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-cyclohexyl-N3-(2-methylpropyl)-4-oxo-N5-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4S)-4-amino-N-ethyl-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}pyrrolidine-2-carboxamide
4-(4-chlorophenyl)-1-[2-(1H-pyrazol-1-yl)ethyl]piperidin-4-ol
3-{2-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
1-cyclopentyl-N3-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
6-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
4-[5-methyl-2-oxo-4-(quinolin-6-ylmethyl)piperazin-1-yl]benzonitrile
N-(3-methylbutyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
3-[(3R,4S)-4-(dimethylamino)-1-{[3-(trifluoromethyl)phenyl]carbamoyl}piperidin-3-yl]propanoic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-ethyl-1H-pyrazole-5-carboxamide
2-[N-(1-methylpiperidin-4-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamido]acetic acid
N-methyl-3-[3-({[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)phenyl]propanamide
ethyl 5-{[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}furan-2-carboxylate
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[2-(pyrazin-2-yl)ethyl]pyridin-2-amine
2-methyl-N-(1,4-oxazepan-6-ylmethyl)thieno[3,2-d]pyrimidin-4-amine