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8-[(1-ethenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,5-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]propan-1-one
(2S,4S)-4-amino-N-(propan-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidine-2-carboxamide
5-methyl-1-propyl-N-[3-(pyridin-2-yl)propyl]-1H-pyrazole-4-carboxamide
N-(3-methyl-1-oxo-1-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}butan-2-yl)acetamide
6-fluoro-N-methyl-2-oxo-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl)-5-(propan-2-yl)-1,2-oxazole
8-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(3-methylbutyl)-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine
5-[(4-fluorophenyl)methyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
methyl 6-(3,5-dimethylbenzoyl)-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl(oxan-2-ylmethyl){[1-(piperidin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl}amine
6-[4-(propan-2-yl)piperazin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
2-[(3-phenylpiperazin-1-yl)methyl]quinolin-4-ol
3-{imidazo[1,2-a]pyridin-2-yl}-5-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazole
1-(2-propyl-1,3-thiazole-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
5-(oxolan-2-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]thiophene-2-carboxamide
(3S,4S)-1-[3-(4-hydroxyphenyl)benzoyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
4,6-dimethyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-[2-(2-oxopiperidin-1-yl)acetyl]piperidine-3-carboxamide
2-methoxy-5-{1-[(3-methylpyridin-2-yl)methyl]-1H-imidazol-2-yl}pyrimidine
N-[(2S)-oxolan-2-ylmethyl]-5-phenyl-1H-pyrazole-3-carboxamide
benzyl 4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carboxylate
4-(5-chloro-2-methoxyphenyl)-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-2-yl)propan-1-one
2-[2-(1H-pyrazol-1-yl)ethyl]-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
2-{1-cyclopentyl-4-[(2,6-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(2-{4-[5-(furan-3-yl)-4-(4-methylphenyl)pyrimidin-2-yl]piperazin-1-yl}ethyl)dimethylamine
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-(cycloheptylamino)-N,N-diethylpyrrolidine-2-carboxamide
N-[2-(2-fluorophenyl)ethyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
1-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)piperidine-4-carboxamide
5-cyclobutyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-1,3,4-oxadiazol-2-amine
1-[2-(4-fluorophenoxy)ethyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-ethyl-4-methyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1,3-thiazole-5-carboxamide
N,N-dimethyl-1-(2-methylpropyl)-5-[(2-phenylethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(1H-imidazol-4-ylmethyl)piperidine-3-carboxylate
2-amino-6-(1H-indol-3-yl)-4-[2-(methoxymethyl)pyrimidin-5-yl]pyridine-3-carbonitrile
N-[(1S,2R)-2-(hydroxymethyl)cyclopentyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
4-[4-(pyrazin-2-yl)piperazin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
N-[(3-methoxyphenyl)methyl]-N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
dimethyl({[4-methyl-5-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
3-(azepane-1-carbonyl)-1-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,5R)-6-methyl-3-(1-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-3-[methyl({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl})amino]propanamide
N-(2-methoxyethyl)-4-({[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)benzamide
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(4-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one