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4-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)pyrimidine
N-(3-cyano-4-methoxyphenyl)-2-(dimethylamino)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
4-(4-{1H,7H-imidazo[4,5-f]indazol-6-yl}-1H-1,2,3-triazol-1-yl)piperidine
2-methyl-N-{2-[methyl(phenyl)amino]propyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
1-ethyl-N-[(5-methylfuran-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4R)-4-amino-1-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide
8-(1-methyl-1H-pyrrole-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(1H-imidazol-2-ylmethyl)-N,2-dimethyl-5-(propan-2-yl)furan-3-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-2-hydroxy-4-methylquinoline-6-sulfonamide
N-benzyl-3-[1-(4-cyanopyridin-2-yl)piperidin-4-yl]-N-methylpropanamide
N-(furan-2-ylmethyl)-9-methoxy-7-oxo-3-[(4-oxo-4H-chromen-3-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2S)-N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-5-(hydroxymethyl)furan-2-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-methoxyethan-1-one
N3-[(4-fluorophenyl)methyl]-N3-(2-methoxyethyl)-N1,N1-dimethylpiperidine-1,3-dicarboxamide
(2S,4S)-1-benzyl-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-chloro-6-methoxy-4-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}phenyl acetate
(3aR,6aR)-2-(2H-1,3-benzodioxole-5-carbonyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-methoxyphenyl)-5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
2-[(3S,4R)-3-cyclopropyl-4-(1-propyl-1H-pyrazole-4-sulfonamido)pyrrolidin-1-yl]acetamide
2-(2,5-dimethylphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
3-[(3R,4S)-1-[2-amino-6-(dimethylamino)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N,N-dimethyl-7-(3-methylbenzoyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3,3-diethyl-1-{[(3S,4S)-3-hydroxy-1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]methyl}urea
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-(3-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(4-fluorobenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(morpholin-4-yl)-2-(4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxy)ethan-1-one
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
(3S,4S)-4-propyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidine-3-carboxylic acid
({1-[(1-cycloheptanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)dimethylamine
(1R,3S)-3-{4-[(4-tert-butylphenyl)methyl]piperazine-1-carbonyl}cyclopentane-1-carboxylic acid
1-[(3aS,6aS)-1-[(4-chloro-3-fluorophenyl)methyl]-octahydropyrrolo[2,3-c]pyrrole-5-carbonyl]-4-methylpiperazine
2-benzyl-9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
8-[(2-ethylpyrimidin-5-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-methyl-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-N-(oxolan-3-ylmethyl)piperidin-4-amine
4-chloro-3-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carbonyl)-1H-pyrazol-5-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,3-benzothiazol-2-yl)piperidin-3-ol
5-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
9-(2-methylbenzoyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-(1-methyl-1H-1,3-benzodiazol-5-yl)urea
1-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-(2-fluoro-4-methylphenyl)-4-phenyl-1H-imidazole
N2-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-N4,6-dimethylpyrimidine-2,4-diamine
4-[(5-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-methylpiperidine
3-hydroxy-3-{[(2-methoxyethyl)(methyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]quinolin-8-ol
N-benzyl-N-methyl-3-[1-(1-phenylcyclopropanecarbonyl)piperidin-4-yl]propanamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-1-(2-methoxyacetyl)piperidine-4-carboxamide