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4-(1H-1,3-benzodiazol-1-yl)-1-(3-methylfuran-2-carbonyl)piperidine-4-carboxylic acid
4-(3-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}piperidin-1-yl)-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-[2-(1H-indol-1-yl)ethyl]propanamide
2-(4-chlorophenyl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
8-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
N-ethyl-1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidine-3-carboxamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
N-[1-(pyrazin-2-yl)propan-2-yl]-1H-1,2,3-benzotriazole-5-carboxamide
methyl 2-[4-(2,3-dihydro-1-benzofuran-5-carbonyl)-2-oxopiperazin-1-yl]acetate
(2E)-N-[2-(2-acetylphenyl)phenyl]but-2-enamide
5-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}-2-(3-methylphenyl)pyrimidine
5-fluoro-N4,N4-dimethyl-N2-[1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-(ethylamino)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrimidine-5-carboxamide
2-(methylsulfanyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1,3-thiazole-4-carboxamide
5-acetyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]thiophene-2-carboxamide
4-(1-{1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-yl}ethyl)morpholine
2-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-fluoro-1-methyl-1H-indole
2-{[4-(3-methylphenyl)-5-[(propan-2-yloxy)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}cyclopropanamine
2-{1-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
4-{[2-(2-fluorophenyl)ethyl]amino}-5-methyl-N-[2-(pyridin-3-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
(2S,4R)-4-amino-N-methyl-1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]pyrrolidine-2-carboxamide
N-(2-hydroxyethyl)-8-oxo-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-ethyl-3,5-dimethyl-1H-pyrazole-4-carboxamide
4-(2-oxo-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-1-yl)benzonitrile
{4-[(4-methoxyphenyl)methyl]-1-[3-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl}methanol
N-(1H-imidazol-2-ylmethyl)-4-[(oxolan-3-yl)sulfamoyl]benzamide
4-{[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-2,3-dihydro-1H-pyrazol-3-one
{1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}methanol
4-[2-(4-methylphenoxymethyl)furan-3-carbonyl]morpholine-2-carboxylic acid
N-(1-methyl-1H-pyrazol-5-yl)-2-{3-[(E)-2-phenylethenyl]-1H-indazol-1-yl}acetamide
7-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
4-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1,4-oxazepane
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[(1R,2S)-2-phenylcyclohexyl]urea
1-[3-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-3-oxopropyl]-1,2-dihydropyridin-2-one
6-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}azocane
5-cyclobutyl-N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1,3,4-oxadiazol-2-amine
2-{2-[3-(benzyloxy)azetidin-1-yl]-2-oxoethyl}-8-methyl-2,8-diazaspiro[4.5]decan-3-one
N-(2-{7-[2-(pyridin-2-ylsulfanyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
N-(2-methylphenyl)-2-{2-[4-(methylsulfamoyl)phenyl]-1H-imidazol-1-yl}acetamide
1-[4-({[2-(furan-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-amino-N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}pyridine-4-carboxamide
1-(methoxymethyl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)cyclobutane-1-carboxamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide