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8-(1-ethyl-1H-pyrazole-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
5-(2-fluorophenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-[(3-methoxyphenyl)methyl]piperidine
1-(2,5-dimethylpyrimidin-4-yl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylic acid
4-{[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-2-yl]methyl}morpholine
1-ethyl-6-methyl-3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{5-[(2-oxo-1,2-dihydropyridin-1-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
6-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-9H-purin-2-amine
1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-3-methyl-3-phenylpiperidine
1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
2-{2-[(4-acetyl-1,4-diazepan-1-yl)methyl]phenyl}-6-methyl-3,4-dihydropyrimidin-4-one
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(pyridin-3-yl)pyridine-3-carboxamide
2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-6-methyl-4-(trifluoromethyl)pyridine
4-[1-(butan-2-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-phenyl-1H-pyrazole
N,N-dimethyl-6-{2-oxa-7-azaspiro[4.5]decan-7-yl}pyrazin-2-amine
N-[2-(diethylamino)ethyl]-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
1-[(2R)-oxolane-2-carbonyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-cyclohexyl-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N3-[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]-N1-(pyridin-3-yl)propane-1,3-diamine
(4S,4aS,8aS)-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
1-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-3-(2-methanesulfonamidoethyl)urea
4-(3-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}propoxy)benzamide
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
1-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(4-sulfamoylphenyl)methyl]propanamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
1-{4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}-1H-imidazole
1-[2-methoxy-5-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrazine-2-carboxamide
(1R,2R,6S,7S)-4-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
ethyl 4-[({1-oxaspiro[4.4]nonan-3-yl}carbamoyl)amino]benzoate
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]propanamide
({4-[(2,6-dimethoxyphenyl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
2-(3-methyl-1-benzofuran-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(pyridin-4-ylmethyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(2-{3-[(4-methoxyphenyl)methyl]-1-methyl-1H-1,2,4-triazol-5-yl}ethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(4-methanesulfonylphenyl)-1-methyl-1H-imidazole
3-(1-methyl-1H-pyrazol-5-yl)-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]propan-1-one
3-(4-fluorophenyl)-N-methyl-3-phenyl-N-(pyridin-2-ylmethyl)propanamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]pyridine-2-carboxamide
ethyl 2-[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]-1,3-oxazole-4-carboxylate
N-(2-methoxyethyl)-15-methyl-13-oxo-9-(pyridin-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
8-methoxy-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(1-phenylpiperidin-4-yl)piperidin-4-ol
(2S,4S)-4-amino-1-(2-fluoro-6-methoxybenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-tert-butyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
4-chloro-2-methoxy-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
2-methoxy-1-{1'-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one