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7-chloro-3-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}quinolin-4-ol
5-fluoro-2-[1-(pyridin-4-ylmethyl)piperidin-2-yl]-1H-1,3-benzodiazole
4-phenyl-3-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine
8-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[1-(4-aminopyrimidin-2-yl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
N-cyclopentyl-4-[4-(2-ethylphenyl)piperazin-1-yl]-4-oxobutanamide
2-(4-acetyl-1,4-diazepan-1-yl)-2-(3-hydroxyphenyl)acetic acid
2-{1-[(2-fluorophenyl)methyl]-4-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
2-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]pyrrolidine-1-carboxamide
N-[1-(thian-4-yl)piperidin-4-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-cyclopropyl-9-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-hydroxy-2-methylpropan-2-yl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-(2-methylprop-2-en-1-yl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
2-(2-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
3-{1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
4-ethyl-5-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1,3-thiazol-2-amine
N-butyl-1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
N-[3-chloro-4-(2,2-dimethylpropanamido)phenyl]-2-acetamido-3-methylbutanamide
2-oxo-8-[(3-phenoxyphenyl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
N-methyl-2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide
2-(2-chloro-4-fluorophenyl)-5-(pyrrolidin-1-ylmethyl)pyridine
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-(ethylamino)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidine-5-carboxamide
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
(3S)-3-{5-[5-(hydroxymethyl)furan-2-yl]-4-phenyl-1H-imidazol-1-yl}azepan-2-one
2-({[(3R,4R)-1-(4-chloro-3-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
8-(2,2-dimethylpropyl)-3-ethyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
4-benzyl-1-(2-butoxyacetyl)-3-ethyl-1,4-diazepan-5-one
2-(2,2-diphenylethyl)-N,N-dimethylmorpholine-4-sulfonamide
5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazole
5-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-2-methylpyridine
[(3R,4R)-1-{[3-(methylsulfanyl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-{3-[5-(azepan-1-ylmethyl)-2-methoxyphenoxy]propyl}-4-(trifluoromethyl)benzamide
3-(azocan-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylpropanamide
2-[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-[(2-methoxyphenyl)methyl]acetamide
1-[2-(1H-imidazol-1-yl)ethyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
4-[5-(1-propylpiperidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]morpholine
1-[1-(1-methyl-1H-imidazol-2-yl)butyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
N-[2-oxo-2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethyl]methanesulfonamide
2-{[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazol-3-yl]formamido}acetamide
2-(2-methoxyphenyl)-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{3-cyclopropyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2,1,3-benzoxadiazole
1-[benzyl(methyl)amino]-3-(5-{[(cyclopropylmethyl)(propyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
5-methoxy-2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenol
5-methoxy-1-methyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-indole-2-carboxamide