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2-[1-(1-benzofuran-3-carbonyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
1-[(3R)-3-cyclopropyl-3-hydroxy-4,4-dimethylpyrrolidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-(2-hydroxyethyl)-8-(quinoxaline-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}quinoline
(3S,5S)-1-(1-benzofuran-2-ylmethyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-[(3R,4S)-4-(dimethylamino)-1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl]propan-1-ol
(3R,5S)-N3-(4-fluorophenyl)-N5-[(3-fluorophenyl)methyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N-cyclopropyl-3,6-dimethyl-N-(thiophen-3-ylmethyl)-1-benzofuran-2-carboxamide
1-{2-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
7-chloro-N,3,5-trimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-benzofuran-2-carboxamide
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}pent-4-enamide
3-(2-methoxy-5-methylphenyl)-6-(2-methoxyphenyl)pyridazine
1-[(1-propyl-1H-imidazol-2-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
1-({[1-(pyrazin-2-yl)piperidin-4-yl]carbamoyl}methyl)piperidine-4-carboxamide
1-(furan-2-ylmethyl)-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]piperidine
(2S)-N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-5-oxopyrrolidine-2-carboxamide
(3S,4S)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(naphthalen-2-yl)piperidin-3-ol
(4aS,7aR)-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,6aR)-2-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-methyl-4-(thiomorpholine-4-carbonyl)-1,2-dihydroquinolin-2-one
(3R,4R)-4-(azepan-1-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-ol
4-[(4-fluoro-3-methylphenyl)methyl]-3-propylmorpholine
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
(1R,2S,9R)-11-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyrrolidin-1-yl)pyridine
4-{4-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]piperazin-1-yl}-2-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
[2-fluoro-5-(5-methyl-1H-indazol-3-yl)phenyl]methanol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
(3S,9aR)-3-(propan-2-yl)-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aR)-6-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
3-{[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}pyridine
methyl({2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})[(2,4,5-trimethoxyphenyl)methyl]amine
2-{[(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
1-cyclopropanecarbonyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]piperidine-4-carboxamide
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
4-ethyl-3-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
N-methyl-2-[methyl(2-phenylethyl)amino]-N-(1H-pyrazol-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
3-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
[(3R,5R)-5-[(dimethylamino)methyl]-1-(2-ethylpyrimidine-5-carbonyl)piperidin-3-yl]methanol
4-(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
N-(pyridin-3-yl)-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)furan-2-carboxamide
4-benzyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-ol
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-(3-methoxypyrazin-2-yl)-4-(pyridin-3-ylmethyl)-1,4-diazepane