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(3S,4S)-1-(4-cyclopentylpyrimidin-2-yl)-4-[(dimethylamino)methyl]piperidin-3-ol
1-(2-amino-2-methylpropyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-(3-chloro-4-propanamidophenyl)quinoline-4-carboxamide
N-cyclopropyl-N-ethyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
7-chloro-N-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
3-[(3R,4S)-1-[3-(dimethylamino)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-methylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[3-(morpholin-4-yl)propyl]acetamide
1-(3-methoxypropyl)-3,8-bis(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-cyclopentyl-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
(3aR,6aS)-2-ethyl-1-oxo-5-[2-(1H-1,2,4-triazol-1-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)piperidine-4-carboxamide
(1R,5R)-N,N-dimethyl-6-(4-phenylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[4-(furan-2-yl)butan-2-yl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
[(3S,5R)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N-cyclopropyl-1-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-ethyl-1-[3-oxo-3-(pyrrolidin-1-yl)propyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]benzoic acid
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(3-methoxyphenyl)piperazine
(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)(2-methylpropyl)(pyridin-2-ylmethyl)amine
1-{[5-(1-ethylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
4-{3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
1-(2,2-dimethyloxan-4-yl)-3-(2-ethyl-6-methylphenyl)-1-methylurea
8-[(4-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
(1S,5R)-6-(2-methoxypyridine-3-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]morpholine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(pyridin-3-yloxy)propyl]benzamide
(1-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}-2-phenylethyl)(methyl)(pyridin-3-ylmethyl)amine
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-ethyl-2-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,3-thiazole-4-carboxamide
N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-(thiophen-3-yl)propanamide
8-[4-(4-hydroxyphenyl)butan-2-yl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N2-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
2-(3-fluorophenyl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
6-(hydroxymethyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}pyridine-2-carboxamide
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)-1-methylpyrrolidine-3-carboxamide
1-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
4-[(2E)-hex-2-en-1-yl]-3-(2-hydroxyethyl)piperazin-2-one
(1-{5-[(adamantan-1-yl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-yl)methanol
1-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperidin-4-ol
2-(2H-1,3-benzodioxol-5-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
2-{[3-(2-methylphenyl)piperidin-1-yl]methyl}pyridine
3-{4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-oxo-1,3-oxazolidine-4-carboxamide
(2S,4S)-N-[2-(2-fluorophenyl)ethyl]-4-[(1-methylpiperidin-4-yl)amino]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
1-cyclohexyl-4-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}piperazine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
5-cyclopropanecarbonyl-1'-[(3-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[1-(2,4-difluorophenyl)ethyl]-4-methylpyrimidin-2-amine
9-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one