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5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(2,4,6-trimethylphenyl)methyl]-1H-pyrazole-3-carboxamide
(1S,5R)-6-benzyl-3-(3-chlorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methoxy-N-methyl-N-(oxan-2-ylmethyl)pyridine-3-carboxamide
4-[(4-acetylpiperazin-1-yl)methyl]-6,8-dimethyl-2H-chromen-2-one
1-[(2-methoxy-5-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]-1H-1,2,4-triazole
N-[4-(1H-indol-2-yl)phenyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
N-{[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
4-[2-(2-phenylethoxy)benzoyl]-1,4-oxazepan-6-ol
1-({5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]furan-2-yl}methyl)pyrrolidine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-phenyl-1H-pyrazole-3-carboxamide
6-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carbonitrile
2-fluoro-N-(oxan-4-yl)-5-sulfamoylbenzamide
methyl 5-[(4-ethylpiperazin-1-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N,N-dimethyl-6-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}pyridine-3-carboxamide
4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-(1-propyl-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanamine
(1R,3S,5S)-8-[4-(5-methylfuran-2-yl)benzoyl]-8-azabicyclo[3.2.1]octan-3-ol
(1s,4s)-4-(4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-1,2,3-triazol-1-yl)cyclohexan-1-amine
2-{2-[(3-cyanopiperidin-1-yl)methyl]phenoxy}acetic acid
2-{4-[(3-fluoropyridin-4-yl)methyl]piperazin-1-yl}-4,6-dimethoxypyrimidine
N,2,5,7-tetramethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]quinoline-4-carboxamide
5-amino-3-(2-methoxy-4-methylphenyl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
N-butyl-2-[(3-methoxyphenyl)methyl]morpholine-4-carboxamide
methyl 4-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)benzoate
N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
2-methyl-3-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2,8-diazaspiro[4.5]decane
1-[(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)methyl]-4-ethylpiperazine
(2S,4R)-4-amino-N-ethyl-1-[(2S)-2-(6-methoxynaphthalen-2-yl)propanoyl]pyrrolidine-2-carboxamide
3-{[3-(5-methylfuran-2-yl)-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
2-methyl-8-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
4,6-dimethyl-2-[4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]pyrimidine
(1R,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
5-[benzyl(methyl)amino]-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
5-(1-cyclopentanecarbonylpiperidin-4-yl)-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-{[(4,4-dimethylpentyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
methyl 4-({3-[(trifluoromethyl)sulfanyl]phenyl}carbamoyl)piperazine-1-carboxylate
N-{2-[bis(propan-2-yl)amino]ethyl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)methanesulfonamide
(3aS,6aR)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-methoxy-1-{1'-[2-(methylamino)pyridine-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-[(5-chlorothiophen-2-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
(2S,4S)-4-{[(2-fluorophenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
12-[3-(diethylamino)pyrrolidine-1-carbonyl]-15-methyl-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-[(5-chlorothiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-methoxyphenyl)methyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
6-(piperidin-4-yl)-2-(thiophen-2-ylmethyl)-3,4-dihydropyrimidin-4-one
3-(2-{[6-(methoxymethyl)pyrimidin-4-yl]amino}ethyl)-4-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one