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1'-{imidazo[1,2-a]pyrimidine-2-carbonyl}-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-[(2-fluoro-5-methoxyphenyl)methyl]-6-oxo-N-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
2-(2-fluoro-4,5-dimethoxyphenyl)-1-[2-(oxan-2-yl)ethyl]-1H-imidazole
N-(5-{[cyclopropyl(1,3-thiazol-2-ylmethyl)carbamoyl]amino}-2-fluorophenyl)acetamide
2-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
1-(pyrimidin-2-yl)-4-[6-(thiomorpholin-4-yl)pyridine-3-carbonyl]-1,4-diazepane
7-chloro-9-oxo-N-(4H-1,2,4-triazol-4-yl)-9H-fluorene-1-carboxamide
8-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(3,4-dimethoxyphenyl)methyl]-3H,4H-pyrido[2,3-d]pyrimidin-4-one
[(3R,4R)-1-(2,4-dimethoxybenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[1-(benzenesulfonyl)piperidin-4-yl]-2-ethylpyrimidine-5-carboxamide
{[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amine
N-methyl-2-(morpholin-4-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
(3R,9aR)-8-[(3-fluorophenyl)methyl]-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-6-(2-methylpropyl)pyrimidin-2-amine
2-ethyl-4-(3-methyl-1H-pyrazole-5-carbonyl)-1-(propan-2-yl)piperazine
(3E)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pent-3-en-1-one
2-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]-4-methoxyphenol
(1S,3R)-3-amino-N-{2-[3-(trifluoromethyl)phenyl]ethyl}cyclopentane-1-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}piperidin-2-one
5-methoxy-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4H-pyran-4-one
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]propanamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylacetamide
2-[(2-{[2-(diethylamino)-2-(furan-2-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
7,7-dimethyl-N-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
4-(2-chloro-4-fluorophenyl)-7H-pyrrolo[2,3-d]pyrimidine
N-(cyclobutylmethyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)benzamide
N-(2-hydroxyethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-[(2-methoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pentan-3-yl)acetamide
2-(1,2-benzoxazol-3-yl)-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)acetamide
1-methyl-6-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-indole
9-(oxane-2-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-[N-methyl-1-(2,6,8-trimethylquinolin-4-yl)formamido]butanamide
ethyl 2-{1-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl}acetate
dimethyl({4-[1-(quinoline-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine
(2-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-2-yl}ethyl)dimethylamine
5-[3-(3-fluoro-4-methoxybenzoyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
4-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-(cyclohexylmethyl)pyrrolidin-2-one
2-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-3,5-dimethoxybenzoic acid
5-methoxy-2-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,4-dihydropyridin-4-one
4-[(dimethylamino)methyl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)azepan-4-ol
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-4-phenylbutan-1-one
3-({[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]oxy}methyl)pyridine
2-[2-(dimethylamino)ethyl]-9-(3-methoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
4-(2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carbonyl)-1,4-oxazepan-6-ol
2-(2H-1,3-benzodioxol-5-yl)-5-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
(4aR,7aS)-1-(3-methylbutanoyl)-4-[(3-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione