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4-ethyl-6-(4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrimidine
1-(4-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
2-{4-[4-(cyclopropylcarbamoyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
2-(4-fluorophenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(piperidin-1-yl)acetamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(dimethylamino)acetamide
N,3-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
3-hydroxy-3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
5-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-(pyridin-2-ylmethyl)piperidin-2-one
N-({2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}methyl)propanamide
(5S)-5-({[(5-ethylpyridin-2-yl)methyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-2-one
(3R,4R)-3-cyclopropyl-4-methyl-1-[1-(morpholin-4-yl)cyclohexanecarbonyl]pyrrolidin-3-ol
1-(3,5-difluoro-4-methoxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(4-methoxyphenyl)-2-methyl-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazine
3-(1-methylpiperidin-3-yl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]propanamide
2-(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N'-butyl-N-(5-methyl-1,2-oxazol-3-yl)-N'-[(3-methylthiophen-2-yl)methyl]ethanediamide
2-(ethylamino)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
2-amino-4-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-5-methyl-6-(propan-2-yl)pyridine-3-carbonitrile
3-[(3R,4S)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-2,6-dimethylquinoline
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
1-{2-oxo-2-[4-(thian-4-yl)piperazin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
N-(1-hydroxybutan-2-yl)-1-(4-methoxyphenyl)-N-(pyridin-3-ylmethyl)cyclopropane-1-carboxamide
N-(1-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
(3S,4S)-N-[4-(furan-2-yl)phenyl]-3,4-bis(hydroxymethyl)pyrrolidine-1-carboxamide
2-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
3-(1,2-dimethyl-1H-imidazol-5-yl)-2,4,5-triazatetracyclo[11.4.0.02,6.07,12]heptadeca-1(17),3,5,7,9,11,13,15-octaene
(3R,4R)-3-cyclobutyl-4-methyl-1-[2-(methylamino)pyridine-4-carbonyl]pyrrolidin-3-ol
methyl 4-(methylsulfanyl)-2-{[1-(3-phenylpropyl)-1H-1,2,3-triazol-4-yl]formamido}butanoate
N-[2-(3-phenylpiperidin-1-yl)ethyl]pyrimidin-4-amine
N'-({1-[(4-tert-butylphenyl)methyl]piperidin-3-yl}methyl)ethanediamide
4-(methylamino)-N-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
(3S)-N3-tert-butyl-N2-(3-fluorophenyl)-1,2,3,4-tetrahydroisoquinoline-2,3-dicarboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}cyclobutanecarboxamide
3-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}propanamide
N-[3-(pyridin-4-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
methyl 2-[2,4-dioxo-1-(2-phenylethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-[(3R,4S)-1-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-4-cyclopropylpyrrolidin-3-yl]methanesulfonamide
2-(2-methoxypyridin-3-yl)-6-(piperidine-1-carbonyl)pyrazine
3-{5-[(5-methylfuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
5,5-dimethyl-3-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-oxazolidine-2,4-dione
5-benzyl-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-[3-(benzenesulfonyl)propanoyl]-1-phenylpiperazin-2-one
N-(3-hydroxy-3-phenylpropyl)-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
(2E)-3-(3-fluorophenyl)-1-{4-[3-(morpholin-4-ylmethyl)phenoxy]piperidin-1-yl}prop-2-en-1-one
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-(1,4-oxazepan-6-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide