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N-(oxolan-2-ylmethyl)-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-propylurea
4-[5-(2-propyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-(oxolan-2-ylmethoxy)ethan-1-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[2-(pyridin-2-ylmethoxy)phenyl]propanamide
6-[3-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-benzothiazole
6-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-3-methyl-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-(4-methoxy-3,5-dimethylbenzoyl)piperidine
N-[2-(diethylamino)ethyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(2-chlorophenyl)methyl]-1-cyclohexanecarbonylpyrrolidine-2-carboxamide
N-(1,2-oxazol-3-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-[(2-fluorophenyl)formamido]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-hydroxypropyl)-3-methoxybenzamide
2-(4-{5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
1-(4-fluorophenyl)-3-methyl-5-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-yl}-1H-1,2,4-triazole
2-[(3,5-difluorophenyl)methyl]-8-(oxolane-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(1-methyl-1H-imidazol-5-yl)methyl]-3-(3-methylphenyl)piperidine
3-(methylsulfanyl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
2-methoxyethyl 7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxylate
4-[(1H-imidazol-2-ylmethyl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
6-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)pyrrolidin-3-yl]methanol
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(1H-imidazol-2-ylmethyl)amino]methyl}piperidin-2-one
1-[(4aS,8aS)-7-cyclopentanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}oxane-2-carboxamide
({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(methyl)[2-(oxan-2-yl)ethyl]amine
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
3-(3-chlorobenzoyl)-1-[(2,5-dimethoxyphenyl)methyl]piperidine
N'1-benzyl-N'1-(1,3-thiazol-2-ylmethyl)cyclopropane-1,1-dicarboxamide
1-{2-[4-(4-ethoxypiperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperazine
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)(thiophen-2-ylmethyl)amine
3-[3-(1H-imidazol-2-yl)propyl]-1-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]urea
(1S,5R)-3-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 2-[4-({[(1r,4r)-4-hydroxycyclohexyl]carbamoyl}amino)phenyl]acetate
1-cyclohexyl-3-methyl-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazole
3-(dimethyl-1,2-oxazol-4-yl)-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
(3S,4R)-4-(4-fluorophenyl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
1-{2-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]phenyl}ethan-1-one
2-(2-methoxyethyl)-8-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-5-{[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]methyl}pyrimidin-2-amine
6-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-[4-({[(3-chlorophenyl)methyl](methyl)amino}methyl)phenyl]-6-methyl-3,4-dihydropyrimidin-4-one
N-(2-{[2-(2-aminoethyl)quinazolin-4-yl]amino}ethyl)acetamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-[(2-methoxyethyl)sulfamoyl]-5-[3-(1H-pyrazol-1-yl)phenyl]benzoic acid
2-(5-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N-(1-methyl-1H-pyrazol-4-yl)-3-({methyl[1-(pyridin-3-yl)propyl]amino}methyl)benzamide