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N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-(propan-2-yl)-1,3-thiazole
2-{1-[(2-methylphenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(3-cyclopentylpropyl)-N-methyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
9-ethyl-1-methyl-4-{2-methylthieno[2,3-d]pyrimidin-4-yl}-1,4,9-triazaspiro[5.6]dodecan-10-one
8-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-(4-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}benzamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
1-(1-cyclohexanecarbonylpiperidin-4-yl)-N-[2-(dimethylamino)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]piperazine-1-carbaldehyde
1-(oxan-4-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]piperidine-3-carboxamide
5-[1-(2-aminoacetyl)pyrrolidin-2-yl]-N-[2-(3-methylthiophen-2-yl)ethyl]thiophene-2-carboxamide
4-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-yl)pyrimidine
1-{2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}pyrrolidin-2-one
5-[1-(2-cyclohexylethyl)-1H-1,2,3-triazol-4-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
2-(3-chloropyridin-2-yl)-2,7-diazaspiro[4.5]decane
5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-4-methylpyrimidin-2-amine
3-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(furan-2-yl)-5-{[3-(3-methylphenyl)piperidin-1-yl]methyl}pyrimidine
N-({5-[(3-fluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
3-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)butanamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(1H-pyrrol-1-yl)ethyl]propanamide
5-[(1,3-benzothiazol-2-ylmethyl)amino]-N-benzyl-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(2-hydroxy-2-phenylpropanoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-(1,3-benzothiazol-2-yl)-4-[(3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-benzyl-4-(4-chlorophenoxy)piperidine-4-carboxamide
3-(2-methylpropyl)-4-{[1-(piperidin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl}morpholine
[(3R,4R)-1-[6-(methoxymethyl)pyridine-2-carbonyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(1-methoxypropan-2-yl)piperidine
3-[1-(propan-2-yl)-1H-pyrazol-5-yl]-1-[3-(pyridin-3-yl)propyl]urea
1-[(2-fluorophenyl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-{[6-(methoxymethyl)pyrimidin-4-yl]amino}ethyl)methanesulfonamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(propan-2-ylsulfanyl)acetamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
5-ethyl-4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-oxazole
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-methylimidazo[1,2-a]pyridine-2-carboxamide
1-phenyl-4-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine
2-({[(3R,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(3R,4S)-4-(3-methoxyphenyl)-1-[3-(prop-2-en-1-yloxy)benzoyl]pyrrolidin-3-amine
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-2-(pyridin-3-yl)acetamide
N-benzyl-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-5-methyl-4-phenyl-1H-imidazole
3-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}-2H-chromen-2-one
3-[(4-methoxyphenyl)methyl]-8-(1-methoxypropan-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(furan-3-ylmethyl)-5-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
8-methoxy-2-[(3-phenoxyazetidin-1-yl)methyl]quinoline
1,3-dimethyl-2,6-dioxo-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide