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({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)[1-(3-methylpyridin-2-yl)ethyl]amine
N-tert-butyl-6-oxo-2-(propan-2-yl)-N-(thiophen-3-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
2-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}benzoic acid
3-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-(3-fluoropyridin-2-yl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
8-[3-(benzyloxy)propyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-3-(1-benzyl-1H-pyrazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
9-(2-methoxypropanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(2-methylphenoxy)piperidin-1-yl]-2-(4-methylpiperazin-1-yl)propan-1-one
1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(2-hydroxy-3-methylbenzoyl)pyrrolidine-2-carboxamide
N-[4-(1H-indol-2-yl)phenyl]-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
5-methyl-N4-[2-(propane-2-sulfonyl)ethyl]pyrimidine-2,4-diamine
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
4-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(furan-2-ylmethyl)-N-methylpiperidine-3-carboxamide
2-(3-methoxypropyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
2-(1-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}pyrrolidin-2-yl)pyridine
(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
5-{4-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]phenoxy}-1H-1,2,3,4-tetrazole
3-{[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}adamantan-1-ol
3-fluoro-2-methoxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
1-butyl-4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperazin-2-one
N4-ethyl-N2-methyl-N2-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
2-amino-7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-(4-phenoxybutyl)-2,8-diazaspiro[4.5]decan-3-one
ethyl 4-{[3-(3-methoxyphenyl)phenyl]carbamoyl}piperidine-1-carboxylate
6-(2H-1,3-benzodioxole-5-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-[1-(2-aminoacetyl)piperidin-4-yl]-N-benzylpiperidine-3-carboxamide
N-({5-[(3-chloro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
methyl 5-(quinoline-8-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-3-methyl-3-phenylbutan-1-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-[({imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)methyl]piperidin-2-one
2-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-1,3-thiazole
1-({4-methyl-5-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
2-amino-4-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{1-[(3-chloro-4-fluorophenyl)methyl]pyrrolidin-3-yl}benzoic acid
1-cyclopropanecarbonyl-N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]piperidine-4-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-benzylpiperidine-4-carboxylic acid
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}-2-phenylacetic acid
5-{[4-(2,4-dimethoxy-3-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}-4-methyl-1,2,3-thiadiazole
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
phenyl (7R,9aR)-7-[(1S)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
1-{1'-[(2S)-1-acetylpyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine