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methyl 3-benzamido-5-({[1-(4-chlorophenyl)cyclopropyl]formamido}methyl)benzoate
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(2-oxo-2-phenylacetyl)piperidine-4-carboxamide
ethyl 3-{[(2H-1,3-benzodioxol-5-yl)carbamoyl]amino}azepane-1-carboxylate
[(3R,4R)-1-(2-methyl-6-propylpyrimidin-4-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-methyl-2-phenyl-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazine
(2S,4S,5R)-5-(2-fluorophenyl)-4-[(furan-3-ylmethyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-5-yl)-2-(2,3-dihydro-1H-inden-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-ethyl-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-4-methyl-1,3-oxazole-5-carboxamide
3-[3-(furan-2-yl)-1-propyl-1H-1,2,4-triazol-5-yl]propanamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
5-(2,6-dimethoxyphenyl)-N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-triazin-3-amine
N-[2-(3-methylthiophen-2-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2,3-dimethyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}quinoxaline-6-carboxamide
4-(5-chloronaphthalene-1-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
2-(2-chlorophenyl)-N-[3-(1H-imidazol-1-yl)propyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
ethyl 4-(cyclopropylmethyl)-1-[4-(1H-indol-3-yl)butan-2-yl]piperidine-4-carboxylate
N-cyclopropyl-N-({4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)-2,3-dimethyl-1H-indole-5-carboxamide
2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
N5,N5,N6-trimethyl-N6-(pyrimidin-4-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[(4-chlorophenyl)methyl]-5-fluoro-N-(3-hydroxypropyl)-1-methyl-1H-indole-2-carboxamide
1-(1,3-benzothiazol-2-ylmethyl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-hydroxy-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyridine-2-carboxamide
8-chloro-2-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
9-(2-oxoimidazolidine-4-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2,2-dimethylpropyl)-4-{[(3-hydroxyphenyl)methyl]amino}pyrrolidin-2-one
5-methyl-N-{3-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}pyridin-2-amine
2-({[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)-6-methoxyphenol
1-{[3-(methylsulfanyl)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-cyclopropyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
({4-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1,3-thiazol-2-yl}methyl)dimethylamine
2-(2-oxopiperidin-1-yl)-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)acetamide
N-[(2-ethoxyphenyl)methyl]-N-ethyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
4-{4-[(4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-ylmethyl}-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-hydroxy-3-methylbenzamide
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2-(4-phenylpiperidin-1-yl)acetamide
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)cyclobutanecarboxamide
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-5-methyl-1H-indazole-3-carboxamide
1-{1-methyl-4-[3-(methylsulfanyl)butyl]-1,4,9-triazaspiro[5.5]undecan-9-yl}pentan-1-one
7-cyclohexyl-2-{[2-(ethylamino)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N,1-dimethyl-N-[2-phenyl-1-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-[5-(thiomorpholin-4-ylmethyl)-1,3-thiazol-2-yl]morpholine
1-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}piperidine-3-carboxamide
3-{5-[(5-acetylthiophen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-N-(2-methyl-1-benzofuran-7-yl)morpholine-4-carboxamide
1-[3-({6-[2-(hydroxymethyl)piperidine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-yl}amino)propyl]pyrrolidin-2-one
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(2-{[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol