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N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]urea
ethyl 4-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}piperidine-1-carboxylate
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-{1-[2-(1H-indazol-1-yl)acetyl]pyrrolidin-2-yl}-N,N-dimethylthiophene-2-carboxamide
3-ethyl-8-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(aminomethyl)phenyl]-4-(3-phenylpropyl)-1,4-diazepane-1-carboxamide
1-(2-{1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-methanesulfonyl-1'-[(3-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-({1-[3-(3-methoxyphenyl)phenyl]piperidin-4-yl}amino)propanamide
N-methyl-5-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
(2E)-3-(2-chlorophenyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)prop-2-enamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
(3R,4R)-3-cyclobutyl-4-methyl-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-3-ol
2-(furan-2-yl)-N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)-2-oxoacetamide
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]methanol
2-(2-chloro-6-fluorophenyl)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-(1H-pyrazol-5-ylmethyl)-1,2-oxazole-3-carboxamide
2-[(3-methyl-1-benzofuran-2-yl)methyl]-2,8-diazaspiro[4.5]decane
N-[(3R,4S)-1-acetyl-4-phenylpyrrolidin-3-yl]-4-sulfamoylbutanamide
(3S,4R)-4-phenyl-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
1-(2,3-difluoro-4-methoxybenzoyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
1-{2-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-benzyl-N,N-dimethyl-5-{[3-(pyridin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-2-(morpholin-3-yl)acetamide
benzyl({3-[3-methyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]propyl})amine
8-(3-ethyl-1,2-oxazole-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}piperidine-3,4-diol
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(1H-pyrazol-1-yl)butanamide
1-(carbamoylmethyl)-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
methyl 4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}butanoate
N-{5-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]pyridin-2-yl}methanesulfonamide
5-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-{imidazo[2,1-b][1,3]thiazol-6-yl}-1,2,4-oxadiazole
4-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-1-ethyl-1H-pyrazole
7-(1,3-benzothiazol-2-yl)-4-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(furan-3-carbonyl)piperidin-3-yl]propanamide
5-ethyl-N-(prop-2-en-1-yl)-N-(propan-2-yl)thiophene-3-carboxamide
2-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-(1-benzylpiperidine-2-carbonyl)piperazin-1-yl]pyrazine
5-{[4-(benzyloxy)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
4-{[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]methyl}benzamide
8-[(3-hydroxyphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(dimethylamino)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-methylpropanamide
7-chloro-4-(oxolan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4S)-4-amino-1-(3-chloro-5-methoxybenzoyl)-N-methylpyrrolidine-2-carboxamide