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methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
1-[3-(pyridin-2-yl)azetidin-1-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
4-cyclobutyl-6-methyl-N-[1-(3-methylpyridin-2-yl)ethyl]pyrimidin-2-amine
(4S)-1-(1H-indol-5-ylmethyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
(3aR,6aS)-5-[(2-hydroxy-7-methylquinolin-3-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(2-chlorophenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-{3-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]piperidin-1-yl}pyrimidine
3-butyl-1-methyl-4-(1H-pyrazole-4-carbonyl)piperazin-2-one
8-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-pyrazole-4-carboxamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3-methylpentane-1,2-dione
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2,3-dihydro-1-benzofuran-5-carboxamide
2-methyl-1-{3-[3-(6-methyl-2-propylpyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
8-methyl-4-[3-(morpholin-4-yl)pyrrolidine-1-carbonyl]-2-(1H-pyrazol-4-yl)quinoline
5-[(4-benzylpiperidin-1-yl)methyl]-N,N-bis(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-4-[(2-methylphenyl)methyl]piperazine
8-(5-fluoropyridine-3-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
7-(cyclopropylmethyl)-2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(thian-4-yl)piperazine
3-acetamido-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}propanamide
1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
6-[(diethylamino)methyl]-N-(2-oxopyrrolidin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
({5-[1-(3-fluoropyridin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
4-[(2S)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carbonyl]morpholine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
3-(2-ethylbutyl)-8-(1-propyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-cyclohexylethyl)-3-hydroxy-3-{[(2-phenylethyl)amino]methyl}piperidin-2-one
N-(2-methoxyethyl)-N,5-dimethyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}pentan-1-ol
1-(2,5-dimethylfuran-3-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
ethyl 4-[({2-[(2-chloroprop-2-en-1-yl)oxy]-6,7-dimethoxyquinolin-3-yl}methyl)amino]piperidine-1-carboxylate
1-{2-[1-(6-chloroquinolin-2-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
4-(4-chlorophenyl)-1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}butan-1-one
N-[(4-fluorophenyl)methyl]-8-methyl-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydroquinoline-3-carboxamide
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
3-{[(4-methanesulfonylphenyl)methyl](methyl)amino}-N-methylbutanamide
(1S,5R)-6-[1-(4-methylphenyl)cyclopropanecarbonyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
N-[2-(oxan-2-yl)ethyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
4-(4-methanesulfonylphenyl)-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-1,2,3-triazole
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,6-dimethyl-1,2-dihydropyridin-2-one
N-cyclopropyl-4-(1H-pyrazol-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
4-(2,3,4-trimethoxyphenyl)-1H-pyrazole-3-carbonitrile
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
(3S,4R)-1-cyclobutanecarbonyl-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-(benzenesulfonyl)-4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide