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1-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
(2S,4R)-N,N-diethyl-4-(2-hydroxybenzamido)-1-propanoylpyrrolidine-2-carboxamide
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-2,3-dihydro-1H-inden-2-amine
4-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)pyrimidin-2-amine
1-{2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydroquinolin-2-one
6-{[4-(3-methylpiperidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
N-[3-(3-methoxyphenyl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
8-[(2R,4S)-4-hydroxypyrrolidine-2-carbonyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-phenoxyethyl)piperidin-3-yl)methanol
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(4-methyl-1,4-diazepan-1-yl)propan-1-one
3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
(2S)-2-({4-[(diethylamino)methyl]-5-ethylfuran-2-yl}formamido)-4-methylpentanamide
1-(cyclopentylmethyl)-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2,4-dimethyl-N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)pyrimidine-5-carboxamide
1-[(4-fluorophenyl)methyl]-4-[2-(methylamino)pyridine-3-carbonyl]piperazin-2-one
(R)-cyclohexyl({3-[2-(methylsulfanyl)ethyl]-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl})methanol
5-{3-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1,3,4-thiadiazol-2-amine
2-(2-hydroxyethyl)-9-(morpholine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-ethoxy-3-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
(4aS,7aR)-1-(3-cyclopropylpropanoyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1-methyl-1H-imidazole-2-carbonyl)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidine
2-{4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}acetamide
5-oxo-1-(pyridin-4-ylmethyl)-N-(thiophen-2-ylmethyl)pyrrolidine-3-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethan-1-one
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
6-fluoro-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
3-benzyl-8-(butan-2-yl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{3-[4-(benzyloxy)piperidin-1-yl]-3-oxopropyl}-5-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-(1-ethoxypropyl)-4-(propan-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]({[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
2-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrazine
3-methyl-N-{3-[2-(2-oxopyrrolidin-1-yl)acetamido]phenyl}benzamide
9-(4-chloro-3-methylbenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[(5-methylpyrazin-2-yl)methyl]-9-(piperidin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-({8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}methyl)pyridin-2-amine
3-{3-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]phenyl}-2,5-dimethylpyrazine
(2S,4R)-4-amino-N-(propan-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
1-(4-fluorophenyl)-2,2-dimethyl-N-[(2-methylpyridin-4-yl)methyl]cyclopropane-1-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2,6-difluorophenyl)methyl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-[4-(4-cyanophenyl)-3-oxopiperazin-1-yl]propanoic acid
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(3-methoxypiperidine-1-carbonyl)-6-(2-methylpropyl)pyrimidin-2-amine
N-benzyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 5-(2,2-diphenylethyl)-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(1,3-benzothiazol-6-yl)-3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]urea
1-ethyl-N-methyl-N-[1-(pyridin-3-yl)pentyl]-1H-pyrazole-3-carboxamide