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4-(4-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine-1-carbonyl)pyridine
1-(3-{4-[(4-methylpentan-2-yl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]acetamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(5-ethylpyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]propanamide
N-(1-{1-[3-(4-fluorophenyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-[3-(1H-imidazol-1-yl)propyl]-1-(pyridin-3-ylmethyl)urea
2-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-methylquinoline
(4aS,7aR)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,1,3-trimethyl-N-[1-(pyridin-3-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(1-benzyl-4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
(3R,5S)-N3-[(5-ethylpyridin-2-yl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
5-(2-methoxypyridin-3-yl)pyridine-3-carboxamide
2-(1-ethyl-1H-pyrazol-4-yl)-3,6-dimethyl-4-(3-methylpiperidine-1-carbonyl)quinoline
N-[4-(1H-imidazol-1-yl)phenyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1,3-oxazole
2,6-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}quinoline-4-carboxamide
2-(1-benzofuran-2-yl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
2-(morpholin-4-yl)-1-[2-(2-phenylethyl)piperidin-1-yl]ethan-1-one
N-methyl-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
4-methanesulfonyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
1-{[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-3-ol
3-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)pyrrolidine-1-carboxamide
6-[3-(1H-pyrazol-1-yl)azetidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
(2R)-2-amino-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-phenylethan-1-one
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-[2-methoxy-5-(morpholin-4-ylmethyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
{1-[(1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
1-{[2-({[2-(2-aminoethyl)quinazolin-4-yl]amino}methyl)phenyl]methyl}pyrrolidin-2-one
1-[(4-chloro-2-fluorophenyl)methyl]-4-cyclopentyl-1,4-diazepane
5-(3-fluorophenyl)-3-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]-1,2,4-triazine
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyrazin-2-amine
7-methyl-2-(morpholin-4-yl)-3-{[2-(trifluoromethyl)morpholin-4-yl]methyl}quinoline
N-{2-[4-oxo-7-(trifluoromethyl)-3,4-dihydroquinazolin-3-yl]ethyl}acetamide
1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}butane-1,2-dione
(5S)-4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,2,2,5-tetramethylpiperazine
3-ethyl-5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-4-methyl-1H-pyrazole
2-amino-8-[3-(1H-pyrazol-1-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-methyl-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-amine
3-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
N-methyl-N-[2-(oxan-4-yl)ethyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
N-(1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidin-3-yl)acetamide
1-cyclopentanecarbonyl-3-[4-(trifluoromethyl)benzoyl]piperidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
5-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-ethyl-N,4-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,3-oxazole-5-carboxamide