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3-[5-(1-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
methyl 4-(4-{4-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)pentanoate
3-(butan-2-yl)-1-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}urea
methyl 3-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-5-(cyclobutylmethoxy)benzoate
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-propylpiperidine
2-[5-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-(carbamoylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
4-chloro-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-ethyl-1H-pyrazole-5-carboxamide
{4-[(4-methoxyphenyl)methyl]-1-(quinoxalin-2-yl)piperidin-4-yl}methanol
4-chloro-N-(1-cycloheptylpiperidin-3-yl)-2-fluorobenzamide
4-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
1-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(5-methylfuran-2-yl)-1H-imidazole
ethyl 2-(1-{2-[4-(2-phenoxyacetamido)-1H-pyrazol-1-yl]acetamido}cyclohexyl)acetate
1-(1-cyclopropanecarbonylpiperidin-4-yl)-2-(phenoxymethyl)-1H-1,3-benzodiazole
N,3-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-(3-chloro-2-fluorophenyl)-3-(hydroxymethyl)-4-methylpiperazine-1-carboxamide
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
N-ethyl-2-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrrole-3-carboxamide
3-methyl-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]benzamide
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(1,3-thiazole-5-carbonyl)piperazine
1-(1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)propan-1-one
(2S,4S)-N-ethyl-1-[(3-methylthiophen-2-yl)methyl]-4-(3,3,3-trifluoropropanamido)pyrrolidine-2-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-5-(propan-2-yl)furan-3-carboxamide
(1s,4s)-N1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}cyclohexane-1,4-diamine
1-[(2-methoxypyridin-3-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one
2-methyl-4-[4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenyl]but-3-yn-2-ol
(4aS,7aR)-6,6-dioxo-4-(2-phenylethyl)-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)butan-1-one
(1R,5R)-6-(cyclobutylmethyl)-3-(5-fluoropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(2-fluorophenyl)methoxy]-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidine
8-methyl-2-propyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-ethyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-6-oxopiperidine-3-carboxamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
5,6-dimethyl-3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(3R,4S)-1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-phenylpyrrolidin-3-amine
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-{[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]amino}-N-(1,3-thiazol-2-yl)propanamide
9-(cyclopropylmethyl)-4-(6-ethyl-2-methylpyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[3-(1H-indazol-1-yl)propyl]-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
4-{6-[4-(pyridin-3-yloxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
5-(4-chloro-1H-pyrazol-3-yl)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-[3,5-difluoro-4-(trifluoromethyl)phenyl]-3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]urea
5-(methoxymethyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[3-(methylsulfanyl)propyl]acetamide
5-chloro-2-(1,4-diazepane-1-carbonyl)-3-phenyl-1H-indole
4-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
N-[(3S)-1-benzylpiperidin-3-yl]-5-ethylpyrimidin-2-amine
2-amino-N-[3-(4-ethoxyphenyl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide