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2-(2-{[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-cyclobutanecarbonyl-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carboxamide
1-[(2-ethyl-5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}furan-3-yl)methyl]pyrrolidine
2,4-dimethyl-5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-thiazole
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxy-2-methylpropan-1-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1,4-dithiepan-6-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]azepane-4-carboxamide
dimethyl[2-({1-[2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}oxy)ethyl]amine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,5-dimethoxybenzamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
methyl 2-(azocane-1-sulfonyl)-6-(4,4,4-trifluorobutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1S,5R)-6-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
7-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2,3,4,9-tetrahydro-1H-carbazole
2-methoxy-4-[(1E)-3-(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)prop-1-en-1-yl]phenol
(2R,3R)-3-[4-(3-hydroxyphenyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-fluoro-2-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-indole
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(2-cyclopentyl-2-phenylacetyl)-1,4-diazepan-5-one
1-benzyl-5-(diethylamino)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-benzyl-3-(1-ethyl-1H-pyrazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(1H-1,3-benzodiazol-2-ylmethyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}amine
N-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)thiophene-2-carboxamide
N-(2-methoxyethyl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-propyl-1H-pyrazole-3-carboxamide
2-[(cyclopropylmethyl)sulfanyl]-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-{2-oxo-4-[2-(pyridin-2-ylsulfanyl)propanoyl]piperazin-1-yl}benzonitrile
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
3-[1-(2-hydroxyacetyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzonitrile
{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
2-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]-5-ethylpyridine
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(thiophen-2-ylmethyl)piperidine
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propan-1-one
N-{[2-(2,3-dimethoxyphenyl)phenyl]methyl}propanamide
2-(morpholin-4-yl)-1-{4-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-(piperidin-4-yl)pyridin-2-amine
1-(2-methyl-5-propylpyrimidin-4-yl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylic acid
4-(3-chloro-4-methoxyphenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-3,5-dimethylbenzamide
3-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1-methyl-1H-indole
1-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-2,4,6-trimethylphenyl)ethan-1-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
4-[(2,2-dimethyloxan-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-(3,4-dichlorophenyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)morpholine