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[(3R,4R)-4-[(dimethylamino)methyl]-1-(quinoline-6-carbonyl)pyrrolidin-3-yl]methanol
5-(1-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)-2-(pyrrolidin-1-yl)pyrimidine
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(cyclopropylmethyl)pyrimidin-2-amine
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-methyl-3-(6-oxo-1,6-dihydropyridazin-3-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
4-[(2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidine-2-carbonyl]morpholine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]pyridine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-(3-hydroxy-1,2-oxazol-5-yl)propanamide
3-[2-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]-5-methylpyridine
4-hydroxy-N-(oxolan-2-ylmethyl)-2-phenylpyrimidine-5-carboxamide
4-{[2-(2-ethylpyrimidin-4-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-3-(thiophen-3-yl)propan-1-one
(butan-2-yl)(3-phenylprop-2-yn-1-yl)(pyridin-2-ylmethyl)amine
5-ethyl-N-methyl-N-[(1-methylpiperidin-4-yl)methyl]pyrimidin-2-amine
5-{[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-[2-(3,5-dimethoxyphenyl)ethyl]-6-(1-methylpiperidin-4-yl)pyrimidin-4-amine
2-(3-fluoropyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazine
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine
4-(2-fluoro-4-methoxyphenyl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
5-chloro-N-[(1r,4r)-4-hydroxycyclohexyl]furan-2-carboxamide
1-(carbamoylmethyl)-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-4-carboxamide
5-{3-[3-(benzyloxy)piperidin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
2-fluoro-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]benzene-1-sulfonamide
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(2-phenylpropyl)piperidine
2-[2-(pyridin-2-yl)ethyl]-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-(1-ethyl-1H-imidazol-2-yl)-1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidine
N-cyclopropyl-2-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}pyridine-4-carboxamide
2-(pyridin-3-yl)-5-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]pyrimidine
4'-[2-(4-chlorophenoxy)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-cyclopropyl-4-methoxy-3-{[1-(3-phenylpropyl)piperidin-4-yl]oxy}benzamide
3-chloro-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}pyridin-2-amine
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,6-dimethylquinoline
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
4-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
4-[4-({[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl)amino}methyl)phenyl]-2-methylbutan-2-ol
4-(2H-1,3-benzodioxol-5-yl)-6-(propan-2-yloxy)pyrimidin-2-amine
N-[(2S,4R,6S)-2-benzyl-6-(4-methoxy-2,5-dimethylphenyl)oxan-4-yl]acetamide
3-{2-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-[4-(propan-2-yl)phenyl]ethan-1-one
(3S,4S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(piperidin-1-yl)pyrrolidin-3-ol
2-tert-butyl-4-hydroxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
3-[(dimethylamino)methyl]-4-(naphthalen-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]propanamide
6-(4-methoxyphenyl)-N-(1-methoxypropan-2-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[phenyl(pyridin-4-yl)methyl]propanamide
2-(4-{3-oxo-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepine-6-carbonyl}piperidin-1-yl)acetamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-[cyclopentyl(methyl)amino]ethan-1-one