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3-(2,5-dimethoxyphenyl)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidine
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-3-phenylpropan-1-one
7-fluoro-2-methyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]quinoline-4-carboxamide
N-(3-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-oxopropyl)acetamide
2-[1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
1-{6-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]pyridin-3-yl}ethan-1-one
(2S,4R)-4-[(cyclohexylmethyl)amino]-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
[(3R,4S)-1-[(3-chlorophenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
1-(2-hydroxyethyl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
3-[4-(aminomethyl)phenyl]-5-(cyclopentylsulfamoyl)benzoic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-[(3-chloro-2-fluorophenyl)methyl]-1,4-oxazepan-5-one
2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-{3-[(3-chlorophenyl)methyl]-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
4-cyclobutaneamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
2-(3-methoxyphenoxy)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
3-[5-(1-benzothiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-({1-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]piperidin-4-yl}methyl)acetamide
4-ethyl-1-[(4-methylbenzenesulfonyl)methyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{5-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[(3-chloro-2-fluorophenyl)methyl]-3-methoxy-2,2-dimethylpropanamide
5-fluoro-N,N-dimethyl-2-[4-(1H-pyrazol-3-yl)piperidin-1-yl]pyrimidin-4-amine
4,6-dimethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(4-propanoylphenoxy)acetamide
N-methyl-3-(5-methylfuran-2-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-[(3-chlorophenyl)methyl]-3-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}propanamide
8-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-benzyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-1H-pyrazole-4-carboxamide
4,5-dimethyl-6-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)pyrimidine
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-ethyl-5-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-(2,3-difluorophenyl)-3-[(4-methanesulfonylmorpholin-2-yl)methyl]urea
3-(1H-imidazol-1-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-1-carboxamide
N6-benzyl-N5-methyl-N5-(oxan-4-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-cyclopropyl-1-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)piperidine-3-carboxamide
N,N-dimethyl-5-(quinolin-4-ylmethyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(1,4-dimethylpiperidin-4-yl)methyl][(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
4-[4-(oxolane-3-carbonyl)piperazin-1-yl]quinazoline
4-(3-methylpiperidin-1-yl)-3-[2-(1H-pyrazol-1-yl)benzamido]benzamide
1-ethyl-4,6-dimethyl-2-oxo-N-[2-(pyridin-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
5-methyl-N4-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidine-2,4-diamine
1-(1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}pyrrolidin-3-yl)-4-methylpiperazine
3-(4-cyano-2-ethylphenyl)-1-[(3R)-piperidin-3-yl]urea
N-(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)acetamide
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
3-(3-methoxypropyl)-1-[2-(trifluoromethyl)benzoyl]piperidine