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1-(2,4-dichlorophenyl)-3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
(2S,4S)-4-amino-N,1-dimethyl-N-(quinolin-6-ylmethyl)pyrrolidine-2-carboxamide
3,5-difluoro-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyridine-2-carboxamide
2-{[(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)oxy]methyl}pyridine
N-ethyl-3-{[4-(thiomorpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
(1S,6R)-9-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(diphenylmethyl)piperazine
5-chloro-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2,3-dihydro-1H-indole-2-carboxamide
methyl 4-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}benzoate
N-methyl-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxamide
{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(2-methylpyridin-4-yl)methyl]amine
2-(2,3-dimethoxy-5-methylphenyl)-2-{methyl[(3-methylpyridin-4-yl)methyl]amino}acetic acid
2-{4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4,6-dimethylpyrimidin-2-amine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-propoxyethan-1-one
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
1-(2-methoxyphenyl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
[(3R,4R)-1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-tert-butyl-3-(ethylamino)-5-(4-methyl-1,4-diazepane-1-carbonyl)benzene-1-sulfonamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
4-{6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carbonyl}-1-phenylpiperazin-2-one
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(furan-2-ylmethyl)(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
5-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-2-cyclopropylpyrimidin-4-ol
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]propan-1-one
2-{4-[2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
3-[(3R,4S)-4-(dimethylamino)-1-(5-methoxy-1H-indole-2-carbonyl)piperidin-3-yl]propanoic acid
3-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
(1R,3s,6r,8S)-4-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
6,7-dimethoxy-2-(3-methoxyphenyl)-3-(1,4-oxazepan-4-ylmethyl)quinoline
2-methyl-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1,3,4-thiadiazole
2-(3-ethoxypropanoyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
7-(1,3-benzothiazol-2-yl)-4-[(4-methoxy-2,5-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
2-(2,2-dimethylpropanoyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[(2S)-pyrrolidin-2-ylmethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amine
1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
1-cycloheptyl-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}oxolane-3-carboxamide
3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-[(1-benzylpiperidin-4-yl)methyl]-N,2,4-trimethylpyrimidine-5-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyridine-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
(1S,5R)-3-(9H-fluoren-2-ylmethyl)-3,9-diazabicyclo[3.3.2]decan-10-one
methyl(oxan-2-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
3-(3,4-dimethoxybenzoyl)-1-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine
N,N-dimethyl-7-(3-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{3-[(3-chlorophenyl)methyl]-5-{[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl}ethan-1-ol