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3-(2-ethyl-1H-imidazol-1-yl)-N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}propanamide
2-(pyridin-3-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrimidine-5-carboxamide
3-(methoxymethyl)-1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-[2-(2-methylphenoxy)ethyl]acetamide
6-[4-(4-methoxyphenoxy)piperidin-1-yl]-N4,N4-dimethylpyrimidine-2,4-diamine
3-(3-hydroxy-3-methylbutyl)-N-[(2-methylpyridin-4-yl)methyl]benzamide
N-{[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]methyl}acetamide
(2R,3S,6R)-5-cyclobutanecarbonyl-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(cycloheptylamino)-2-methylheptan-2-ol
2-[3-(2-methylpropyl)-1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
4-[hydroxy(pyridin-2-yl)methyl]-N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)piperidine-1-carboxamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-{4-[(pyridin-2-yl)amino]piperidin-1-yl}propan-1-one
N-(4-acetylphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
3,5-dimethyl-1-(1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}pyrrolidin-3-yl)-1H-pyrazole
{[5-(4-ethoxyphenyl)furan-2-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-methylpiperidine-2-carboxamide
2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]-N-cyclopentyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
N-(adamantan-2-ylmethyl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-dimethyl-5-(1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-{[(3-methyloxetan-3-yl)methyl]sulfamoyl}benzamide
(4aR,7aS)-1-(2-methylpropyl)-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[(3R,5S)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)-N,4-dimethylpiperazine-1-carboxamide
6-ethyl-4-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}-1,2-dihydropyridin-2-one
5-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
[1-(2,8-dimethylquinoline-4-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-(cyclopent-1-en-1-yl)-1-{4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
3-(3-chlorophenyl)-N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
(2R,3S,6R)-3-phenyl-5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1-methyl-1H-1,2,3-benzotriazole
(2R,6R)-4-[(3-ethyl-1,2-oxazol-5-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{2-[bis(propan-2-yl)amino]ethyl}-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)furan-3-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
3-benzyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperazin-2-one
N-methyl-N-(1H-pyrazol-5-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
5-({[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-N,N-dimethylpyrimidin-2-amine
6-{3-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
5-acetyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]thiophene-2-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-methyl-6-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(dimethylamino)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
(1S,5R)-3-(3-fluoropyridin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-fluoro-5-methylphenyl)-3-{[(1R,2S)-2-(methoxymethyl)cyclopentyl]amino}propanamide
6-ethyl-N,N-dimethyl-2-[2-(2-methylpropyl)pyrimidin-5-yl]quinoline-4-carboxamide
N-{3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-4-methylbenzamide
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]urea