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N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-hydroxy-1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-[3-(5-fluoro-2-methylphenyl)phenyl]-2-methoxyacetamide
1-cyclohexyl-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
4-[5-cyclopropyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
N-(7-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N'-(4-methylphenyl)propanediamide
2-[(4-chlorophenyl)methyl]-8-[3-(dimethylamino)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(2S)-2-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
2-amino-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
1-(2-methylpropyl)-4-oxo-N3-(propan-2-yl)-N5-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3,5-dicarboxamide
({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amine
(3S,4R)-1-(1-benzofuran-5-ylmethyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
1-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
4-{[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]methyl}benzoic acid
2-(3-fluoro-4-methylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
2-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidine
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
8-(2-aminopyrimidin-4-yl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(1H-indazol-1-yl)propyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
N-methyl-3-(quinolin-8-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-2-ylmethyl)benzamide
2-[2-(2-oxopyrrolidin-1-yl)ethyl]-N-(2-phenylethyl)piperidine-1-carboxamide
(4aS,7aR)-1-(4-chloro-2-fluorobenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[3-(2-oxopiperidin-1-yl)propanoyl]piperidine-3-carboxylate
ethyl 1-(1,4-dithiepan-6-yl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
3-(3-fluorophenyl)-N-{1-oxaspiro[4.5]decan-3-yl}-1H-pyrazole-4-carboxamide
5-(3,3-diphenylpiperidine-1-carbonyl)-1,2-dihydropyridin-2-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
8-(5-methyl-1,2-oxazole-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-ethyl-3-(1-methyl-1H-1,2,3-triazol-4-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]urea
1-(1,4-dioxan-2-ylmethyl)-2-(4-methoxynaphthalen-1-yl)-1H-imidazole
4-(2,6-dimethylpyridin-3-yl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methylpyrimidin-2-amine
4-(1-butyl-1H-imidazol-2-yl)-1-(pyrrolidine-1-sulfonyl)piperidine
(3R,5S)-N-[(3,4-dimethoxyphenyl)methyl]-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-amine
1-cyclopropyl-5-{[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
4-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1-methylpyrrolidin-2-one
N-{[6-(2,3-difluorophenyl)pyridin-3-yl]methyl}acetamide
N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)quinoline-8-carboxamide
N6-cyclopropyl-N5-methyl-N5-[1-(1,3-thiazol-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-(1-{1-[(3-chloro-1-benzothiophen-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-[2-(4-chlorophenoxy)ethyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
1-(1,3-benzoxazol-2-yl)-N-{1-oxaspiro[4.4]nonan-3-yl}piperidin-4-amine
4-[(2-chloro-4-fluorophenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
3-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-N-[(2-methoxyphenyl)methyl]propanamide
2-(3,4-dimethylpiperazine-1-carbonyl)-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
9-(2,6-difluoro-4-methoxybenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(1R,3S)-7-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol