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N-benzyl-2-[(3-methoxyphenyl)amino]-N-methylbutanamide
(2S,4R)-4-[4-(2-fluoro-4-methylbenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
N-(2-methoxy-6-methylphenyl)-3-[(4-methyl-1,4-diazepan-1-yl)methyl]benzamide
2-(cyclopentylmethyl)-1,6-dimethyl-3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
5-methyl-1-(2-oxo-2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[2-(2,3-dihydro-1H-inden-1-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}azepan-3-amine
2-cyclopropyl-4-phenyl-9-(2-propoxyacetyl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-4-oxo-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[(1S)-1-phenylethyl]-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(4-ethenylphenyl)urea
1-cyclopropyl-5-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidine-3-carboxamide
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-(2-oxopyrrolidin-1-yl)benzamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2S)-pyrrolidine-2-carbonyl]piperidine
[2-(3,5-dimethylphenoxy)ethyl]({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
N-({5-[(2-methylnaphthalen-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
N,N-dimethyl-5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-2-methyl-1,3-oxazole
N-(2-hydroxy-3-methoxypropyl)-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-1λ6-thiomorpholine-1,1-dione
(4aS,7aR)-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[4-({[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)carbamoyl}methoxy)phenyl]propanamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(5-ethylthiophene-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-({1-benzyl-5-[1-(methoxymethyl)cyclobutyl]-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
4-(1H-imidazol-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
2-(1-methylpyrrolidin-3-yl)-9-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-fluorophenoxymethyl)-N-methyl-N-[2-(piperidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-(3-fluoropyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3,4-difluorophenyl)methyl]-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}propanamide
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(4-chlorophenoxy)piperidin-1-yl]propan-1-one
1-methyl-6-(propan-2-yl)-3-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-(cyclopropylmethyl)-5-[5-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-{4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenyl}acetamide
{1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]urea
1-{1-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
3-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-N-(pyridin-3-yl)benzamide
N-ethyl-N-[2-(4-methoxyphenoxy)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
N1-[2-(3-phenylpropoxy)phenyl]piperidine-1,4-dicarboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2R)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
N-[4-(5-methyl-4-{[(1-methylpiperidin-2-yl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-3-carboxamide
2-(3-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}piperidin-1-yl)pyridine
N-(4-fluorophenyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-amine
1-[(3,3-diphenylpiperidin-1-yl)sulfonyl]-4-methylpiperazine
2-(4-{3-methyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
1-[2-(dimethylamino)ethyl]-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide