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({1-[1-(1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)dimethylamine
N-methyl-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-N-(thiophen-3-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[3-(1-methylcyclopropyl)propanoyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-methoxy-N-{8-methyl-2-oxo-4-[2-(prop-2-en-1-yloxy)phenyl]-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}pent-4-enamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-4-sulfamoylbenzamide
1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
1-(4-methyl-2-{[2-(3-phenylpiperidin-1-yl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
1-[2-(pyrrolidin-1-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-phenylethane-1,2-dione
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propane-1,2-dione
5-cyclopropyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
3-(1-methylpiperidin-2-yl)-N-[(6-methylquinolin-5-yl)methyl]propanamide
2-[(1-ethyl-5-oxopyrrolidin-3-yl)amino]-N-[(2-methoxyphenyl)methyl]acetamide
6-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}sulfonyl)-1,2,3,4-tetrahydroquinoxaline-2,3-dione
(3R,4R)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
3-(2-methyl-1H-imidazol-1-yl)-1-[3-(3-methylphenyl)piperidin-1-yl]propan-1-one
3-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzonitrile
1-methyl-2-[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]-1H-1,3-benzodiazole
(2R,3R)-3-{[(4-methoxyphenyl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(2-methoxyethyl)-4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
3-(2-amino-1,3-thiazol-4-yl)-N-[1-(thiophen-3-yl)propan-2-yl]propanamide
1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
2-{2-[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyridazine-3-carboxamide
2-[1-(oxane-2-carbonyl)piperidine-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
[(3R,4R)-1-[3-(dimethylamino)pyrazin-2-yl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
3-(1-methyl-1H-pyrrol-2-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-{[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}acetamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
3-{1-[1-(4-fluorophenyl)cyclopropanecarbonyl]pyrrolidin-2-yl}-4-methyl-1,2,5-oxadiazole
N-(2-methoxyethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2S)-2-(methoxymethyl)-N-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}pyrrolidine-1-carboxamide
2-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)piperidin-1-yl]pyrimidine
N-(adamantan-2-yl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
1-[(3,4-difluorophenyl)methyl]-5-[4-(2,3-dimethylphenyl)piperazin-1-yl]azepan-2-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-fluoro-2-methoxybenzamide
4-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholine
4-cyclopropyl-1-[(4-methoxypyridin-2-yl)methyl]-4-methylpyrrolidin-2-one
4-(3-fluoropyridin-4-yl)-6-methyl-7-(2-oxopyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
(2R)-2-cyclohexyl-1-[4-(ethoxymethyl)piperidin-1-yl]-2-hydroxyethan-1-one
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-5-methyl-N-[(6-methylpyridin-2-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
1-[(4-fluorophenyl)methyl]-4-(1-methyl-1H-imidazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane