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9-(3-ethyl-1,2-oxazole-5-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
5-oxo-1-phenyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2,5-dihydro-1H-pyrazole-3-carboxamide
(2S,4S)-4-amino-1-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-N-methylpyrrolidine-2-carboxamide
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-3-ol
2-(4-{4-[(2,3-dihydroxypropyl)(methyl)amino]pyrimidin-2-yl}piperazin-1-yl)-N-ethylacetamide
2-(2-fluorophenyl)-N-{2-[(2S)-pyrrolidine-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}acetamide
6-ethyl-2-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]quinoline-4-carboxamide
(2S,4R)-1-[(3-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-(pentan-3-yl)-N-(2-phenylethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
N-methyl-2-(1-methyl-1H-imidazol-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
3-{[(4-fluorophenyl)methyl]amino}-N-[(3-methyl-1H-pyrazol-5-yl)methyl]benzamide
5-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-2-cyclohexylpyrimidine
N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-(2-methyl-1-benzofuran-5-carbonyl)-1,2-oxazolidin-4-ol
1-(3-phenylpropyl)-4-(1-propyl-1H-pyrazole-5-carbonyl)-1,4-diazepane
6-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-9H-purin-2-amine
4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-4-ylmethyl)piperazine
1-cyclopentyl-4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
5-[3-(1H-pyrazol-3-yl)phenyl]-1H-indole
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-indazole-3-carboxamide
4-[5-(cyclobutylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
4-[(5-ethylpyridin-2-yl)methyl]-N-(4-fluorophenyl)piperazine-2-carboxamide
N-({1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-3-yl}methyl)-3-(trifluoromethyl)benzamide
5-{2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}pyrrolidin-2-one
4-(4-chlorophenyl)-1-[4-(propan-2-yl)pyrimidin-2-yl]piperidin-4-ol
2,6-dimethyl-4-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)phenyl acetate
[4-(5-propyl-1,3,4-oxadiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
dimethyl[3-({5-[4-(1,3-oxazol-5-yl)phenyl]pyridin-2-yl}oxy)propyl]amine
2-{1-[5-(2-chlorophenyl)furan-2-carbonyl]azetidin-3-yl}pyridine
N-(2-methoxyethyl)-4,6-dimethyl-2-oxo-N-(1,3-thiazol-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-(3-phenylprop-2-ynoyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
8-butyl-N-(2-fluorophenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]pyrrolidin-3-yl]acetamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]benzamide
8-(2-fluoro-6-methoxybenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(2-ethylpyrimidin-4-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
2-methyl-4-[4-(2-phenylazetidine-1-carbonyl)phenyl]butan-2-ol
2-[1-(cyclohexylmethyl)-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl]ethan-1-ol
3-[(1H-imidazol-2-ylmethyl)[(5-methylthiophen-2-yl)methyl]amino]propan-1-ol
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-hexylpiperidine
4-{1-[1-(4-tert-butylbenzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
3-(5-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3,5-dimethyl-N-(propan-2-yl)-1-benzofuran-2-carboxamide
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(1H-indol-3-ylmethyl)methylamine
2-(2-hydroxyethyl)-9-[(3-methylquinoxalin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-acetyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine-2-carboxamide