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3-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}benzonitrile
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
7-fluoro-2-(3-propyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
1-[5-(methoxymethyl)furan-2-carbonyl]-4-{2-[(3-methoxyphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
(2H-1,3-benzodioxol-4-ylmethyl)(butan-2-yl)(pyridin-4-ylmethyl)amine
2-[(3,5-difluorophenyl)methyl]-8-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1,3,5-trimethyl-7-[6-(piperidin-4-yl)pyrimidin-4-yl]-3,7-diazabicyclo[3.3.1]nonane
1-(cyclopent-3-en-1-yl)-5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazole
3,5-dimethyl-4-{1-[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
11-[methyl(1,3-thiazol-4-ylmethyl)amino]-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
7-(5-methylthiophen-2-yl)-4-[2-(1H-pyrazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
4-{2-[2-(trifluoromethoxy)phenyl]pyridine-4-carbonyl}morpholine
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2,1,3-benzoxadiazole
1-[(4-methoxyphenyl)methyl]-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperazin-2-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
7-(2-methoxyphenyl)-2-(2-methylpyridin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(1-hydroxybutan-2-yl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
ethyl 3-[5-(2-cyanophenyl)-4-phenyl-1H-imidazol-1-yl]propanoate
2-[(2-methylprop-2-en-1-yl)oxy]-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)benzamide
1-(oxolane-2-carbonyl)-4-(2,3,5,6-tetramethylbenzoyl)piperazine
(2S)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-{3-[(dimethylamino)methyl]phenyl}-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{4-[1-(3-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
2-{3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
3-({1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-N,N-bis(prop-2-en-1-yl)benzamide
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
(adamantan-1-ylmethyl)({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-ethyl-1H-pyrazole-5-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
2-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-3-carboxamide
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(furan-3-ylmethyl)-1,4-diazepan-6-ol
N-[(3R,4S)-1-(carbamoylmethyl)-4-phenylpyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
N-[5-(2-methanesulfonylacetamido)-2-methoxyphenyl]benzamide
1-methyl-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
2-methyl-5-[4-(oxan-2-ylmethyl)phenyl]-1,3,4-oxadiazole
6-(4-fluorophenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
2-(furan-3-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
9-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methoxyethyl)-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
(3S,4S)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
2-[methyl(2-phenylethyl)amino]-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-3-(2,3-dihydro-1H-isoindol-2-yl)propan-1-one
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4,5-dimethyl-1H-imidazol-1-yl)ethan-1-one
2-({2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)-6-fluoroquinolin-4-ol
1-(cyclohexylmethyl)-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
5-chloro-3-methyl-2-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-indole