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7-(3,6-dimethylpyrazin-2-yl)-4-[(2-ethoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclohexyl-N-(thiophen-3-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[(2-ethoxy-2-oxoethyl)carbamoyl]piperidine-3-carboxylate
4-{5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}-1-phenylpiperazin-2-one
N-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-4-(1H-pyrazol-3-yl)piperidine-1-carboxamide
N-[2-(methylsulfanyl)ethyl]-1-(3-phenylphenyl)piperidin-4-amine
2-(2,3-dihydro-1H-inden-1-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
4-[6-(2-fluoro-6-methoxyphenyl)pyridine-3-carbonyl]morpholine
ethyl 1-{[4-(2-hydroxyethoxy)phenyl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-cyclobutyl-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-(2,5-dimethylphenyl)-3-methyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
1-(4-cyclohexylphenyl)-3-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-3-methylurea
N-[(2-chloropyridin-3-yl)methyl]-6-ethyl-N,2-dimethylquinoline-4-carboxamide
3-benzyl-1-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
8-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]quinoline
1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(4-{[2-(6-ethoxyquinolin-2-yl)-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
5-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-1,2-dihydropyridin-2-one
(2S)-3-phenyl-2-{[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propanamide
4-(4-fluorophenoxy)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperidine
N-{2-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-3-methylpyridin-4-amine
(1R,5R)-3-cyclobutanecarbonyl-6-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
[(5-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)(pyridin-4-ylmethyl)amine
1-[1-(hydroxymethyl)-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-phenylethan-1-one
5-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-8-fluoroquinoline-2-carboxamide
2-(2-{4-[5-(hydroxymethyl)furan-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,2,3,4-tetrahydrophthalazine-1,4-dione
3-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[3-(4-fluorophenyl)phenyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidine-2-carboxamide
N-({1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
1-[2-(1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
3-cyclopropyl-1-(2-methoxyphenyl)-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole
2-amino-N-[2-(dimethylsulfamoyl)ethyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
1-(4-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
2-(cyclopentylmethyl)-6-methyl-1-(pyridin-3-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one
1-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-(5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1H-pyrazol-3-yl)phenol
(2S,4S)-1-cyclopentyl-N,N-diethyl-4-(3-methylthiophene-2-amido)pyrrolidine-2-carboxamide
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
5-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-2-ol
2-[methyl(pyridin-3-ylmethyl)amino]-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)acetamide
7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-[2-(propylsulfanyl)phenyl]-1-[1-(pyridin-4-yl)propan-2-yl]urea
2-(5-acetylthiophen-3-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
(4aS,8aR)-6-[5-(methoxymethyl)furan-2-carbonyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
3-(furan-2-yl)-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-fluoro-2-methoxy-N-[(1-methylpiperidin-3-yl)methyl]benzamide