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N-(4-{[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)carbamoyl}phenyl)-2-methylfuran-3-carboxamide
1-(3-fluoropyridin-4-yl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-acetyl-8-[(4-butoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2-methoxy-5-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
2-(3,4-dichlorophenyl)-4-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)morpholine
N-methyl-N-(oxan-4-yl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-(4-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-({[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
1-benzyl-5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(2R,6R)-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carbonyl)-N,N-diethylpiperidine-3-carboxamide
1-(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-2-methylpropan-1-ol
1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,3,5-trimethylfuran-2-carboxamide
6-[3-(2-fluorophenyl)benzoyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
3-{1-[(3-chloro-4-methoxyphenyl)methyl]piperidin-2-yl}propanoic acid
3-{[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
(1R,5R)-6-benzyl-3-(cyclopropanesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
7-(4-methoxy-3-methylbenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1-(propan-2-yl)piperidin-4-amine
2-[3-(2-methoxyphenyl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
5-(dimethoxy-1,3,5-triazin-2-yl)-1H-indole
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylpropanamide
{1-[(4-ethynylphenyl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
1-{3-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-oxopropyl}piperidin-2-one
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-(pyridin-2-yl)piperidin-4-ol
5-[4-(dimethylamino)naphthalene-1-carbonyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(2-methoxyphenyl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(5-acetylthiophen-3-yl)-N-[2-(4-fluorobenzenesulfonyl)ethyl]acetamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-1-(2,3-dimethylphenyl)piperidin-4-amine
N-{[(2S,4S)-4-fluoro-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl]methyl}pyrrolidine-1-carboxamide
1-{4-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-butyl-N-[(4-fluorophenyl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-N-(2-chlorophenyl)propanamide
(5-{1-[1-(benzenesulfonyl)piperidin-4-yl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-5-(methoxymethyl)furan-2-carboxamide
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
5-[1-(2-chloro-6-fluoro-3-methylbenzoyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
(2R)-N-(1-butyl-4-methyl-1H-pyrazol-5-yl)oxolane-2-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)butanoyl]piperazin-2-one
2-ethoxy-5-[2-(3-hydroxy-3-methylpiperidin-1-yl)pyrimidin-4-yl]benzoic acid
3-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-2,3-dihydro-1λ6-thiophene-1,1-dione
(3S,4R)-4-(4-fluorophenyl)-1-(2-hydroxy-5-methylbenzoyl)pyrrolidine-3-carboxylic acid
(3R,4R)-4-cyclopropyl-1-[3-(2-methoxyphenoxy)propyl]-3-methylpiperidin-4-ol
2-cyclohexyl-2-[1-(2-hydroxyethyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]acetic acid
N-(3-cyclopentylpropyl)-3-(4-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
2-(1H-imidazol-2-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}benzamide
2-(2-hydroxypropanoyl)-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(1H-imidazol-4-ylmethyl)-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane